2 Results for "

NK-2R antagonist

" in MedChemExpress (MCE) Product Catalog:
Products (2)

2 Results for "NK-2R antagonist" in MCE Product Catalog:

Cat. No.: HY-122286
CAS No.: 272104-60-6
Target:  

Neurokinin Receptor

Research Areas:  

Neurological Disease

SB 414240 is a selective neurokinin-2 receptor (NK-2R) antagonist with Kis of 1 nM and 193 nM for human NK-3R and human NK-2R, respectively. SB 414240 does not bind the human μ-opioid receptor (hMOR). SB 414240 can be used for the study of neurological disease .
loading...
    loading...
Cat. No.: HY-117053
CAS No.: 169340-04-9
Target:  

Neurokinin Receptor

Research Areas:  

Neurological Disease

ZM 253270 is a species-selective non-peptide NK-2 receptor (NK-2R) antagonist. ZM 253270 competitively inhibits the binding of [ 3H]NKA to native or cloned NK-2R from hamster bladder (Ki=2 nM), but has a weaker inhibitory effect (48-fold) on the binding of [ 3H]NKA to cloned human NK-2R .
loading...
    loading...