4 Results for "

aromatatase

" in MedChemExpress (MCE) Product Catalog:
Products (4)

4 Results for "aromatatase" in MCE Product Catalog:

Cat. No.: HY-113986
CAS No.: 102676-87-9
Purity:  98.75%
Synonyms: (R)-Fadrozole; (R)-CGS 16949A free base; FAD286
Target:  

Cytochrome P450

Research Areas:  

Cardiovascular Disease

Dexfadrostat ((R)-Fadrozole) is an orally active and selective aromatase inhibitor, with human aromatase IC50 values of 6.4 nM. Dexfadrostat suppresses estrogen synthesis, reduces circulating estradiol levels and suppresses aldosterone production. Dexfadrostat can be used for the research of breast cancer, primary aldosteronism, and hypertension .
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Cat. No.: HY-P11837
Research Areas:  

Cancer

NECT-224 is a bifunctional chelator and a nectin-4 targeting peptide conjugate. NECT-224 can be used as a PET imaging agent when labeled with 64Cu or 68Ga .
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Cat. No.: HY-136745
CAS No.: 331684-05-0
Target:  

Cytochrome P450

Research Areas:  

Cancer

Aromatase-IN-1 is a competitive aromatase (P450arom) inhibitor with a human IC50 of 40 nM and a Ki of 1.05 nM. Aromatase-IN-1 binds via coordination of imidazole nitrogen to the heme iron of aromatase. Aromatase-IN-1 can be used for the research of breast cancer .
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Cat. No.: HY-113986C
CAS No.: 131863-75-7
Synonyms: (R)-Fadrozole hydrochloride; (R)-CGS 16949A; FAD286 hydrochloride
Target:  

Cytochrome P450

Research Areas:  

Cardiovascular Disease Cancer

Dexfadrostat ((R)-Fadrozole) hydrochloride is an orally active and selective aromatase inhibitor, with human aromatase IC50 values of 6.4 nM. Dexfadrostat hydrochloride suppresses estrogen synthesis, reduces circulating estradiol levels and suppresses aldosterone production. Dexfadrostat hydrochloride can be used for the research of breast cancer, primary aldosteronism, and hypertension .
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