34 Results for "

deuterated derivative

" in MedChemExpress (MCE) Product Catalog:
Products (34)

34 Results for "deuterated derivative" in MCE Product Catalog:

Cat. No.: HY-12215S2
CAS No.: 2131126-33-3
Synonyms: PF-06463922-d3-1
Deulorlatinib (compound A), a deuterated derivative of Lorlatinib (HY-12215), is a potent inhibitor of tyrosine kinase demonstrating the potential for the research of ALK-positive advanced NSCLC .
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Cat. No.: HY-116666S
(Rac)-Etomidate acid-d5 is the deuterium labeled (Rac)-Etomidate acid .
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Cat. No.: HY-D0300S1
CAS No.: 1173021-13-0
Leucomalachite green-d6 is the deuterated derivative of Leucomalachite green (HY-D0300). Leucomalachite green is the major reduced metabolite of malachite green (MG) and has lower cytotoxicity (such as HEp-2 and Caco-2) than malachite green. Leucomalachite green may be involved in interfering with cell metabolism or redox balance and can be used to evaluate its potential harm to human cells as a food contaminant .
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Cat. No.: HY-B0007S2
CAS No.: 2012598-58-0
Baclofen-d5 hydrochloride is deuterated labeled Baclofen (HY-B0007). Baclofen, a lipophilic derivative of γ-aminobutyric acid (GABA), is an orally active, selective metabotropic GABAB receptor (GABABR) agonist. Baclofen mimics the action of GABA and produces slow presynaptic inhibition through the GABAB receptor. Baclofen has high blood brain barrier penetrance. Baclofen has the potential for muscle spasticity research .
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Cat. No.: HY-B0661CS
CAS No.: 1189923-88-3
(Rac)-Tamsulosin-d3 hydrochloride is the deuterated-labeled Tamsolusin hydrochloride (HY-B0661C). Tamsolusin hydrochloride (YM12617 hydrochloride; LY253351 hydrochloride) is an isomer of Tamsulosin (HY-B0661). Tamsolusin hydrochloride is a sulfonamide phenethylamine derivative and a competitive antagonist of selective post-synaptic α1-adrenoceptors. Tamsolusin hydrochloride inhibits CYP3A4 activity in a non-competitive, enantiomer-specific manner, with an IC50 and Ki of 6.75 μM. Tamsolusin hydrochloride produces dose-dependent hypotension, preferentially antagonizing α1-adrenoceptor-mediated pressor responses, and inhibits α2-adrenoceptor-mediated pressor responses at high doses. Tamsolusin hydrochloride can be used in research related to various diseases such as metabolism .
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Cat. No.: HY-113404S1
CAS No.: 157929-66-3
L-Dopa-d3 is deuterated labeled DL-Dopa (HY-113404). DL-Dopa is a beta-hydroxylated derivative of phenylalanine.
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Cat. No.: HY-137222S
CAS No.: 1309283-30-4
4',5-Dihydroxy Diclofenac-13C6 is a deuterated derivative of Diclofenac (HY-15036). Diclofenac is a potent COX inhibitor with anti-inflammatory activity .
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Cat. No.: HY-W141927S
CAS No.: 3008541-77-0
N-Heptanoylglycine-d2 is the deuterated labeled N-Heptanoylglycine (HY-W141927). N-Heptanoylglycine is a Glycine (HY-Y0966) derivative .
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Cat. No.: HY-W141934S
CAS No.: 3008541-76-9
N-Valerylglycine-d2 is the deuterated labeled N-Valerylglycine (HY-W141934). N-Valerylglycine is a Glycine (HY-Y0966) derivative .
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Cat. No.: HY-W142395S
6-TAMRA-d12 free acid is a deuterated-labeled 6-TAMRA, which is widely used in the preparation of fluorescent antibodies and as a fluorescent group for immunohistochemical avidin derivatives.
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Cat. No.: HY-10882S1
Clotrimazole-d10 is deuterated labeled Clotrimazole (HY-10882). Clotrimazole is an imidazole derivative, an antifungal compound and is a CYP (cytochrome P450) inhibitor. Clotrimazole has antibacterial activity.
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Cat. No.: HY-W012850S1
DL-Cysteine-d1 is the deuterated labeled 2-Amino-3-mercaptopropanoic acid (HY-W012850). 2-Amino-3-mercaptopropanoic acid is a cysteine derivative .
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Cat. No.: HY-114591S
CAS No.: 2470126-90-8
Spiromesifen-d9 is a deuterated labeled Spiromesifen . Spiromesifen (BSN 2060) is a broad-spectrum tetrachloro acid derivative acaricide. Spiromesifen can interfere with lipid biosynthesis, and has no cross-resistance to any resistant mite or whitefly populations .
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Cat. No.: HY-60351S
CAS No.: 2222933-95-9
5-Aminopyrimidine-d3 is the deuterated form of 5-Aminopyrimidine. 5-Aminopyrimidine is a biochemical reagent that can serve as a biomaterial or an organic compound for research related to life sciences. Its derivatives exhibit antioxidant activity .
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Cat. No.: HY-141749AS
CAS No.: 1217614-64-6
Synonyms: CLPM-d4; SR 26334-d4
Clopidogrel carboxylic acid-d4 is a deuterated derivative of Clopidogrel carboxylic acid, which is an inactive metabolite of the antiplatelet agent Clopidogrel (HY-15283) in plasma. Clopidogrel carboxylic acid-d4 can be used to further explore the metabolic characteristics of Clopidogrel .
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Cat. No.: HY-163591
CAS No.: 3034034-10-8
PRMT5-IN-36-d3 is the deuterated derivative of PRMT5-IN-36. PRMT5-IN-36-d3 (compound 4) is an orally active PRMT5 inhibitor for cancer research .
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Cat. No.: HY-N6710S
CAS No.: 1778734-73-8
α-Zearalenol-d4 is a deuterated labeled α-Zearalenol . α-Zearalenol is a Mycotoxin with high affinity for the estrogen receptors (ER), α-Zearalenol is the derivative of zearalenone (ZEN), causes reproductive disorders in animals, due to its xenoestrogenic effects .
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Cat. No.: HY-168547S
CAS No.: 3021566-15-1
AR89-d6 (Compound AR102) is a deuterated derivative of AR89 with oral activity. AR89-d6 demonstrates activity against S. mansoni, S. haematobium, and S. japonicum, and can be utilized for research on schistosomiasis .
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Cat. No.: HY-125658S
Biotinyl tyramide-d4 is a deuterated labeled Biotinyl tyramide (HY-125658). Biotinyl tyramide is a biotin derivative used for tyramide signal amplification (TSA), as a reagent to amplify both immunohistochemical signals and in situ hybridization protocols. Biotinyl tyramide can be used for the research of tyramide signal amplification .
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Cat. No.: HY-59140S2
(S)-2-Amino-3,3-dimethylbutanoic acid-d6 is a deuterated labeled (S)-2-Amino-3,3-dimethylbutanoic acid . (S)-2-amino-3,3-dimethylbutanoic acid is a leucine derivative .
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