COX Inhibitors

COX

COX-1

COX-2

COX-3

COX Inhibitors, Activators, Modulators & Controls

Product Name	COX	COX-1	COX-2	COX-3	Purity
Acetaminophen		COX-1, IC₅₀: 113.7 μM	COX-2, IC₅₀: 25.8 μM		99.97%
EIPA			COX-2		99.73%
Oxidopamine hydrobromide			COX-2		99.42%
Indomethacin		Human COX-1, IC₅₀: 18 nM (in CHO cells)	Human COX-2, IC₅₀: 26 nM (in CHO cells)		99.90%
Celecoxib		COX-1, IC₅₀: 15 μM	COX-2, IC₅₀: 40 nM		99.89%
4'-Acetoxy resveratrol			COX-2		99.90%
Moracin G			COX-2
Aspirin		COX-1, IC₅₀: 27.75 μM	COX-2, IC₅₀: 1.17 mM		99.90%
Oxidopamine hydrochloride			COX-2		99.91%
Gallic acid			COX-2		99.99%
Diclofenac		Human COX-1, IC₅₀: 4 nM (in CHO cells) Ovine COX-1, IC₅₀: 5.1 μM	Human COX-2, IC₅₀: 1.3 nM (in CHO cells) Ovine COX-2, IC₅₀: 0.84 μM		99.92%
Ibuprofen		COX-1, IC₅₀: 13 μM	COX-2, IC₅₀: 370 μM		99.97%
Catechin		COX-1, IC₅₀: 1.4 μM			99.30%
Sodium propionate			COX-2		99.0%
20(S)-Ginsenoside Rg3			COX-2		99.82%
(-)-Epicatechin		COX-1, IC₅₀: 3.2 μM			99.00%
Meloxicam		COX-1, IC₅₀: 36.6 μM	COX-2, IC₅₀: 0.49 μM		99.59%
Naproxen		COX-1, IC₅₀: 9.55 μM	COX-2, IC₅₀: 5.65 μM		99.98%
Xanthohumol		COX-1	COX-2		99.94%
Salicylic acid			COX-2		98.42%
Diclofenac Sodium		Human COX-1, IC₅₀: 4 nM (in CHO cells) Ovine COX-1, IC₅₀: 5.1 μM	Human COX-2, IC₅₀: 1.3 nM (in CHO cells) Ovine COX-2, IC₅₀: 0.84 μM		99.81%
EIPA hydrochloride			COX-2		98.01%
Ketoprofen		COX-1, IC₅₀: 2 nM (in human blood monocytes)	COX-2, IC₅₀: 26 nM (in human blood monocytes)		99.95%
Carprofen		COX-1, IC₅₀: 22.3 μM	COX-2, IC₅₀: 3.9 μM		99.94%
Rebamipide			COX-2		99.74%
NS-398			COX-2, IC₅₀: 3.8 μM		99.71%
(-)-Epicatechin gallate		COX-1, IC₅₀: 7.5 μM			99.96%
Ginsenoside C-K			COX-2		99.93%
Aspirin (Standard)		COX-1	COX-2
Neochlorogenic acid			COX-2		99.80%
Mefenamic acid		hCOX-1, IC₅₀: 40 nM	hCOX-2, IC₅₀: 3 μM		99.95%
Phenacetin				COX-3, IC₅₀: 102 μM	99.95%
Isoorientin			COX-2, IC₅₀: 39 μM		98.36%
(S)-(+)-Ibuprofen		COX-1, IC₅₀: 2.1 μM	COX-2, IC₅₀: 1.6 μM		99.98%
SC-560		COX-1, IC₅₀: 9 nM	COX-2, IC₅₀: 6.3 μM		99.79%
Sodium Salicylate			COX-2		99.99%
Rutaecarpine		COX-1, IC₅₀: 8.7 μM (in BMMC)	COX-2, IC₅₀: 0.28 μM (in BMMC)		99.09%
Valdecoxib		COX-1, IC₅₀: 140 μM	COX-2, IC₅₀: 5 nM		99.89%
α-Amyrin			COX-2		99.99%
Flurbiprofen	COX	COX-1	COX-2		99.95%
Iguratimod			COX-2, IC₅₀: 20 μM		98.49%
Ibuprofen sodium		COX-1, IC₅₀: 13 μM	COX-2, IC₅₀: 370 μM		99.98%
Piroxicam		COX-1, IC₅₀: 47 μM (in human monocytes)	COX-2, IC₅₀: 25 μM (in human monocytes)		99.78%
Madecassic acid			COX-2		99.93%
Crocetin			COX-2		98.07%
MS-444			COX-2		99.42%
Ginsenoside Rd			COX-2		99.88%
Guaiacol			COX-2		99.96%
Niflumic acid			COX-2, IC₅₀: 100 nM		99.61%
Rofecoxib			Human COX-2, IC₅₀: 18 nM (in Chinese hamster ovary cells) Human COX-2, IC₅₀: 26 nM (in human osteosarcoma cells)		99.89%
Nimesulide			COX-2, IC₅₀: 0.07-70 μM		99.89%
Terameprocol			COX-2		99.50%
Fenofibric acid			COX-2, IC₅₀: 48 μM		99.94%
γ-Tocopherol	Cyclooxygenase				99.63%
Oxaprozin		COX-1, IC₅₀: 2.2 μM	COX-2, IC₅₀: 36 μM		99.94%
Psoralidin			COX-2		99.90%
Sodium thiosulfate (99%, water≤1.0%)			COX-2		99.89%
Gamma-Mangostin			COX-2		99.91%
Naproxen sodium		COX-1, IC₅₀: 9.55 μM (in intact cells )	COX-2, IC₅₀: 5.65 μM (in intact cells )		99.74%
Salicin	COX				99.43%
STAT1/3-IN-1			COX-2
Ethyl Caffeate			COX-2		99.34%
S-(+)-Marmesin			COX-2		99.9%
Corynoline			COX-2		98.84%
Syringaldehyde			COX-2, IC₅₀: 19.2 μM		99.96%
Diflunisal	COX				99.82%
Etoricoxib		COX-1, IC₅₀: 116 μM (in human whole blood)	COX-2, IC₅₀: 1.1 μM (in human whole blood)		99.86%
Isofraxidin			COX-2		99.94%
α-Humulene			COX-2		98.55%
Jaceosidin			COX-2		99.51%
Parecoxib			COX-2		99.29%
Pectolinarigenin			COX-2		99.98%
cis-5-Dodecenoic acid		COX-1	COX-2		99.76%
Sinapaldehyde			COX-2, IC₅₀: 47.8 μM		99.71%
Roburic acid		COX-1, IC₅₀: 5 μM	COX-2, IC₅₀: 9 μM		99.93%
Guluronic acid sodium			COX-2		98.0%
Prim-O-glucosylcimifugin			COX-2		99.87%
Salicylic acid-d₆			COX-2		99.82%
Isobavachin			COX-2		99.88%
Paradol			COX-2		99.87%
Tolfenamic Acid			COX-2, IC₅₀: 13.49 μM (in cell)		99.94%
Harpagoside		COX-1	COX-2		99.88%
Etodolac		COX-1, IC₅₀: ∼50000 nM (in CHO cells)	COX-2, IC₅₀: 41 nM (in CHO cells)		99.48%
Ketorolac		COX-1, IC₅₀: 20 nM	COX-2, IC₅₀: 120 nM		99.87%
Ginsenoside Rg5			COX-2		99.88%
Licofelone	COX, IC₅₀: 0.21 μM				99.84%
Avicularin			COX-2		99.80%
Ginsenoside Rb3			COX-2		99.87%
Macelignan			COX-2		99.85%
Glafenine		COX-1	COX-2		98.77%
Acetaminophen (Standard)		COX-1	COX-2
Lumiracoxib		COX-1, Ki: 3 μM	COX-2, Ki: 0.06 μM		99.93%
Cafestol			COX-2		99.91%
Kukoamine A			COX-2		99.88%
Callistephin chloride			COX-2		98.31%
Nabumetone			COX-2		99.94%
[8]-Shogaol			COX-2, IC₅₀: 17.5 μM		99.93%
Oxatomide			COX-2		98.11%
S-(+)-Ketoprofen		COX-1, IC₅₀: 13 μM	COX-2, IC₅₀: 370 μM		99.88%
Militarine			COX-2		99.94%
Broussonin E			COX-2		98.11%
Fenoprofen Calcium hydrate	COX				99.52%
Parecoxib Sodium			COX-2		99.82%
AG-024322		COX-1, Ki: 2.3 nM	COX-2, Ki: 3 nM		98.27%
Gnetol		COX-1, IC₅₀: 0.78 μM			99.86%
Ketorolac tromethamine salt		COX-1, IC₅₀: 20 nM	COX-2, IC₅₀: 120 nM		99.53%
Lornoxicam		COX-1, IC₅₀: 5 nM (in cells)	COX-2, IC₅₀: 45 nM (in cells)		99.36%
Pranoprofen		COX-1	COX-2		98.56%
3,3'-Diiodo-L-thyronine	COX
Moracin C			COX-2		99.54%
Ecliptasaponin A			COX-2		99.81%
[10]-Shogaol			COX-2, IC₅₀: 7.5 μM		99.78%
Dendrophenol			COX-2		99.93%
Humulone			COX-2		99.46%
Glafenine hydrochloride		COX-1	COX-2		99.03%
Salicylic acid (Standard)			COX-2
SC-236		COX-1, IC₅₀: 17.8 μM	COX-2, IC₅₀: 10 nM		99.59%
Tolmetin		Human COX-1, IC₅₀: 0.35 μM	Human COX-2, IC₅₀: 0.82 μM		99.54%
Loxoprofen		COX-1, IC₅₀: 6.5 μM (in human whole blood)	COX-2, IC₅₀: 13.5 μM (in human whole blood)		99.57%
Inulicin			COX-2		99.94%
Hexahydrocurcumin			COX-2		99.70%
β-Elemonic acid			COX-2		99.77%
DuP-697		hCOX-1, IC₅₀: 800 nM	hCOX-2, IC₅₀: 10 nM		99.79%
(-)-Catechin gallate		COX-1	COX-2		99.98%
Octahydrocurcumin			COX-2		99.25%
(+)-Catechin hydrate		COX-1, IC₅₀: 1.4 μM			99.59%
Geranial			COX-2		99.51%
FK 3311			COX-2		98.72%
N-tert-Butyl-α-phenylnitrone			COX-2		99.94%
Imrecoxib		Human COX-1, IC₅₀: 115 nM	Human COX-2, IC₅₀: 18 nM		99.48%
Regaloside B			COX-2		99.90%
Cornuside			COX-2		99.99%
Triflusal		COX-1			99.56%
Deracoxib			COX-2		99.96%
Gallic acid hydrate			COX-2		99.98%
Anthraquinone-2-carboxylic acid			COX-2		98.0%
Ampyrone	COX				99.72%
Zaltoprofen		COX-1, IC₅₀: 1.3 μM	COX-2, IC₅₀: 0.34 μM		98.89%
Tenoxicam		COX-1	COX-2		99.93%
Flunixin meglumine		COX-1, IC₅₀: 0.55 μM	COX-2, IC₅₀: 3.24 μM		99.65%
NF-κB/MAPK-IN-1			COX-2		98.71%
Edpetiline			COX-2		99.81%
Mofezolac		COX-1, IC₅₀: 1.44 nM	COX-2, IC₅₀: 447 nM		99.34%
Hydralazine			COX-2		99.94%
Phenacetin (Standard)				COX-3
Tenidap		COX-1, IC₅₀: 0.03 μM	COX-2, IC₅₀: 1.2 μM		99.93%
Bromfenac sodium		COX-1, IC₅₀: 5.56 nM	COX-2, IC₅₀: 7.45 nM		99.92%
N-(p-Coumaroyl) Serotonin			COX-2		99.03%
Revaprazan hydrochloride			COX-2		99.98%
Bromfenac sodium hydrate		COX-1, IC₅₀: 5.56 nM	COX-2, IC₅₀: 7.45 nM		99.94%
2,4-Dihydroxybenzaldehyde			COX-2		99.93%
Gynostemma Extract			COX-2		99.92%
3,4-Dihydroxyphenylglycol			COX-2		98.07%
PT109			COX-2		99.20%
Dihydrokavain		COX-1	COX-2		99.94%
Rehmannioside A			COX-2		99.96%
Nepafenac		COX-1, IC₅₀: 64.3 μM	COX-2, IC₅₀: 0.12 μM		99.56%
(-)-Epicatechin gallate (Standard)		COX-1
(-)-Epicatechin (Standard)		COX-1
Saponarin			COX-2		99.95%
BMP-4 (15-24) acetate			COX-2		99.30%
Byakangelicol			COX-2		99.48%
Phenidone	COX				98.96%
Diclofenac acyl glucuronide		COX-1, IC₅₀: 0.620 μM	COX-2, IC₅₀: 2.91 μM		98.34%
Tilmicosin phosphate			COX-2		98.0%
Aceclofenac		COX-1, IC₅₀: 7.3 μM	COX-2, IC₅₀: 3 μM		99.83%
Diclofenac potassium		Human COX-1, IC₅₀: 4 nM (in CHO cells) Ovine COX-1, IC₅₀: 5.1 nM	Human COX-2, IC₅₀: 1.3 nM (in CHO cells) Ovine COX-2, IC₅₀: 0.84 nM		99.85%
2,5-Di-tert-butylhydroquinone			COX-2, IC₅₀: 14.1 μM		99.90%
Fenbufen		COX-1, IC₅₀: 3.9 μM	COX-2, IC₅₀: 8.1 μM		98.50%
(S)-Flurbiprofen		COX-1, IC₅₀: 0.48 μM	COX-2, IC₅₀: 0.47 μM		99.88%
α-Spinasterol		COX-1, IC₅₀: 16.17 μM	COX-2, IC₅₀: 7.76 μM		99.90%
Indobufen	COX				99.98%
(E)-Ethyl p-methoxycinnamate		COX-1, IC₅₀: 1.12 μM	COX-2, IC₅₀: 0.83 μM		99.39%
Phenethyl ferulate	COX, IC₅₀: 4.35 μM				99.66%
α-Chaconine			COX-2		99.76%
CAY10404		COX-1, IC₅₀: >500 μM	COX-2, IC₅₀: 1 nM		99.40%
Pelubiprofen			COX-2		98.46%
Lupeol acetate			COX-2		98.0%
TFAP		COX-1, IC₅₀: 0.8 μM			99.98%
Eicosatetraynoic acid	COX, ID₅₀: 8 μM				99.9%
Phenyl β-D-glucopyranoside			COX-2		99.85%
Asaraldehyde			COX-2		99.42%
2,4-Dinitrobenzenesulfonic acid sodium salt			COX-2		99.98%
PTUPB		COX-1, IC₅₀: 100 μM	COX-2, IC₅₀: 1.26 μM		98.05%
Pheophytin a			COX-2
Felbinac		COX-1, IC₅₀: 865.68 nM	COX-2, IC₅₀: 976 nM		99.94%
SC-58125		hCOX-1, IC₅₀: >100 μM	hCOX-2, IC₅₀: 0.04 μM		99.92%
Columbin		COX-1, EC₅₀: 327 μM	COX-2, EC₅₀: 53.1 μM		99.80%
2′-Hydroxy-5′-methoxyacetophenone			COX-2		99.96%
Timosaponin A1			COX-2, IC₅₀: 36.43 μM		99.70%
Acemetacin		COX-1, IC₅₀: 85 μM (in human intact cell)			99.95%
Diclofenac diethylamine		Human COX-1, IC₅₀: 4 nM (in CHO cells) Ovine COX-1, IC₅₀: 5.1 μM	Human COX-2, IC₅₀: 1.3 nM (in CHO cells) Ovine COX-2, IC₅₀: 0.84 μM		99.95%
Loxoprofen sodium		COX-1, IC₅₀: 6.5 μM	COX-2, IC₅₀: 13.5 μM		99.63%
7,3',4'-Tri-O-methylluteolin			COX-2		99.28%
Hydrangenol			COX-2		99.63%
β-Amyrone			COX-2		99.87%
Sericin			COX-2
Sphondin			COX-2		99.70%
Isoastragaloside I			COX-2		99.49%
Fenofibric acid (Standard)			COX-2
Firocoxib		COX-1, IC₅₀: 7.5 μM	COX-2, IC₅₀: 0.13 μM		99.54%
Vedaprofen		COX-1			98.73%
Ufenamate			COX-2		99.89%
Alminoprofen			COX-2		99.91%
Otenaproxesul		COX-1	COX-2		98.03%
ARN14494			COX-2		99.08%
Darutoside			COX-2		99.89%
Floctafenine		COX-1	COX-2
Iminostilbene			COX-2		99.34%
Madecassic acid (Standard)			COX-2
Casuarinin			COX-2		98.24%
trans-Isoferulic acid			COX-2		99.93%
Alisol F			COX-2		99.89%
Ketorolac-d₅		COX-1, IC₅₀: 20 nM	COX-2, IC₅₀: 120 nM		98.75%
Adelmidrol			COX-2		98.0%
Indazole-Cl			COX-2		98.19%
FR122047		COX-1, IC₅₀: 28 nM			99.55%
Oleocanthal		COX-1	COX-2		≥99.0%
4,4'-Dihydroxy-2,6-dimethoxydihydrochalcone		COX-1	COX-2		99.64%
Flurbiprofen axetil	COX				99.34%
Wnt/β-catenin-IN-6			COX-2		98.34%
Enflicoxib			COX-2		99.88%
Thymohydroquinone			COX-2		99.91%
Plantanone B		Ovine COX-1, IC₅₀: 21.78±0.2 μM	Ovine COX-2, IC₅₀: 44.01±0.42 μM		99.16%
Propyphenazone	COX				99.85%
Tolmetin sodium dihydrate		Human COX-1, IC₅₀: 0.35 μM	Human COX-2, IC₅₀: 0.82 μM		99.94%
2-(p-Tolyl)propanoic acid		COX-1, IC₅₀: 38.23 μM	COX-2, IC₅₀: 64.30 μM
Δ7-Avenasterol			COX-2
Polmacoxib			COX-2, IC₅₀: 0.1 μg/mL		99.70%
Cholesteryl eicosapentaenoate		COX-1, IC₅₀: 14.6 μg/mL	COX-2, IC₅₀: 17.3 μg/mL		99.9%
Phellodendrine			COX-2		99.60%
Dipyrocetyl			COX-2		98.16%
Valeryl salicylate		COX-1			99.0%
Desmethyl Celecoxib			COX-2, IC₅₀: 32 nM		99.42%
Shizukaol B			COX-2
BW 755C		COX-1, IC₅₀: 0.65 μg/mL	COX-2, IC₅₀: 1.2 μg/mL
Oleanolic acid 28-O-β-D-glucopyranoside			COX-2		99.42%
Diplacone			COX-2		98.38%
Benzanthrone			COX-2
15(R)-Lipoxin A4			COX-2		98.3%
Crocetin (Standard)			COX-2
Ocarocoxib			COX-2, IC₅₀: 1.4 μM		99.94%
Tebufelone			COX-2		99.52%
Teriflunomide impurity 3		COX-1, IC₅₀: 30 μM			99.75%
Amfenac Sodium Hydrate			COX-2		98.33%
Nitroaspirin		COX-1			98.57%
Indomethacin-d₄		Human COX-1, IC₅₀: 18 nM (in CHO cells)	Human COX-2, IC₅₀: 26 nM (in CHO cells)		99.78%
Mavacoxib			COX-2		99.04%
(S)-(+)-Ibuprofen-d₃		COX-1, IC₅₀: 2.1 μM	COX-2, IC₅₀: 1.6 μM		99.96%
1-Methyl-6-oxo-1,6-dihydropyridine-3-carboxylic acid			COX-2		99.94%
Pamicogrel	Cyclooxygenase				99.44%
GW-406381			COX-2		99.69%
Anemarsaponin B			COX-2		99.43%
Isoxicam		COX-1	COX-2		99.83%
Hamaudol		COX-1, IC₅₀: 0.3 mM	COX-2, IC₅₀: 0.57 mM		99.98%
Cimicoxib			COX-2		98.02%
3,9-Dihydroeucomin			COX-2
Guluronic acid			COX-2		98.90%
Gaultherin			COX-2, IC₅₀: 250 μg/mL		99.44%
SC57666			COX-2, IC₅₀: 26 nM		98.94%
FR-188582			COX-2, IC₅₀: 17 nM		99.12%
Garcinoic acid			hCOX-2
Isoxicam (Standard)		COX-1	COX-2
Nitroflurbiprofen	COX				99.64%
RWJ 63556			COX-2		99.35%
Ketoprofen (lysinate)		COX-1, IC₅₀: 2 nM	COX-2, IC₅₀: 26 nM
COX-2-IN-6			COX-2		98.80%
Revaprazan			COX-2
Aspirin lithium		COX-1	COX-2
Indomethacin sodium		COX-1, IC₅₀: 18 nM	COX-2, IC₅₀: 26 nM
COX-2-IN-28		COX-1, IC₅₀: 13.21 μM	COX-2, IC₅₀: 0.054 μM
Geiparvarin			COX-2
Tolmetin sodium		Human COX-1, IC₅₀: 0.35 μM	Human COX-2, IC₅₀: 0.82 μM
SD 8381		hCOX-1, IC₅₀: 0.69 μM	hCOX-2, IC₅₀: 0.0098 μM
COX-2-IN-56			COX-2
Jaceosidin (Standard)			COX-2
EGFR-IN-190			COX-2, IC₅₀: 0.208 μM
JNUTS013			COX-2
Daturaolone		COX-1
Antitumor agent-77			COX-2
Brazzein			COX-2, IC₅₀: 12.62 μM
COX-1-IN-1		COX-1, IC₅₀: 0.23 μM	COX-2, IC₅₀: 50 μM
Desmethyl etoricoxib		COX-1, IC₅₀: 16 μM	COX-2, IC₅₀: 1 μM		99.64%
COX-2/LOX-IN-1			COX-2, IC₅₀: 0.55 μM
COX-1/2-IN-2		COX-1, IC₅₀: 9.7±0.09 μM	COX-2, IC₅₀: 4.6±1.45 μM
Topo I/COX-2-IN-2			COX-2, IC₅₀: 2.31 μM
Cassiatannin A			COX-2
TX-1123		COX-1, IC₅₀: 15.7 μM	COX-2, IC₅₀: 1.16 nM
COX-2-IN-21		COX-1, IC₅₀: 12.4 μM	COX-2, IC₅₀: 0.039 μM
Anti-inflammatory agent 110			COX-2
Anti-inflammatory agent 109			COX-2
Longiferone B			COX-2
MAO-B-IN-56			COX-2, IC₅₀: 7.83 μM
COX-2-IN-27		COX-1, IC₅₀: 13.22 μM	COX-2, IC₅₀: 0.045 μM
VU0487836		Ovine COX-1, IC₅₀: 0.36 μM			99.86%
LM-4108		Ovine COX-1, IC₅₀: >66 μM	Human COX-2, IC₅₀: 60 nM
COX-1/2-IN-12		Human COX-1, IC₅₀: 41.6 nM	Human COX-2, IC₅₀: 31.1 nM
Arnicolide B			COX-2
COX-2-IN-5			COX-2, IC₅₀: 0.65 μM
Ginsenoside Rb3 (Standard)			COX-2
ISP-VT			COX-2
G721-0282			COX-2		99.96%
COX-2-IN-17		COX-1, IC₅₀: >10 μM	COX-2, IC₅₀: 0.02 μM
VI-60			COX-2
Ginsenoside C-K (Standard)			COX-2
COX-2/5-LOX-IN-8			Ovine COX-2, IC₅₀: 6.3 μM
COX-2/15-LOX-IN-6			COX-2, IC₅₀: 0.201 μM
Antitumor agent-78			COX-2
COX-2-IN-51			COX-2, IC₅₀: 70.7 nM
EGFR/VEGFR2-IN-11			COX-2, IC₅₀: 17.38 μM
LY256548	Cyclooxygenase
COX-2-IN-65			COX-2, IC₅₀: 10.24 μM
2,5-Dimethoxy-3-glucopyranosylcinnamic alcohol		COX-1
COX-2-IN-58			COX-2
Ginsenoside Rd (Standard)			COX-2
BChE-IN-46			COX-2, IC₅₀: 0.11 μM
EGFR/VEGFR2-IN-10			COX-2, IC₅₀: 158 nM
threo-Guaiacylglycerol β-coniferyl ether		COX-1	COX-2
COX-1-IN-4		COX-1, IC₅₀: 0.09 μM	COX-2, IC₅₀: 2.49 μM
COX-2-IN-47			COX-2, IC₅₀: 0.03 μM
iNOS/COX-2-IN-1			COX-2
Zidometacin		COX-1	COX-2
COX-1/2-IN-1		COX-1, IC₅₀: 9.7±0.09 μM	COX-2, IC₅₀: 4.6±1.45 μM
SIN 14			COX-2
COX-2-IN-46			COX-2, IC₅₀: 87.74 nM
COX-2-IN-31		COX-1, IC₅₀: 12.5 μM	COX-2, IC₅₀: 60 nM
COX-2-IN-10			COX-2
Anti-inflammatory agent 111			COX-2
Ephemeranthol A			COX-2
Clematomandshurica saponin B			COX-2
Kadsulignan N			COX-2
EGFR/COX-2-IN-3			COX-2, IC₅₀: 0.15 μM
Vitacoxib			COX-2
CHNQD-03005			COX-2
COX-2/sEH-IN-1		COX-1, IC₅₀: 8.72 μM	COX-2, IC₅₀: 1.24 μM
Meloxicam sodium		COX-1, IC₅₀: 36.6 μM	COX-2, IC₅₀: 0.49 μM
2,4-Dihydroxybenzaldehyde (Standard)			COX-2
COX-2-IN-60		COX-1, IC₅₀: 5.93 μM	COX-2, IC₅₀: 0.06 μM
COX-2-IN-48			Human COX-2, IC₅₀: 51.7 nM
COX-2-IN-30		COX-1, IC₅₀: 10.4 μM	COX-2, IC₅₀: 49 nM
LYRM03			COX-2
cis-5-Dodecenoic acid (Standard)		COX-1	COX-2
Oxaprozin potassium		COX-1, IC₅₀: 2.2 μM	COX-2, IC₅₀: 36 μM
Taraxerol acetate		COX-1, IC₅₀: 116.3 μM	COX-2, IC₅₀: 94.7 μM		98.0%
COX-2-IN-16			COX-2, IC₅₀: 102 μM
EGFR/COX-2-IN-1		COX-1, IC₅₀: 20.1 μM	COX-2, IC₅₀: 1.52 μM
COX-2-IN-14			COX-2
COX-2/Aromatase-IN-1			COX-2
BPN-37440			COX-2, IC₅₀: 42 nM
1α-Hydroxyvitamin D5			COX-2
Caspase-3/7 activator 4			COX-2, IC₅₀: 5.38 μM
TU-100			COX-2
Parameritannin A-1			COX-2
4F-PMPH			COX-2
Ermanin			COX-2		99.47%
Lefucoxib			COX-2
COX-1/2-IN-3		COX-1	COX-2
Parsalmide		Ovine COX-1, IC₅₀: 9.92 μM	Ovine COX-2, IC₅₀: 155 μM
COX-2/HDAC6-IN-1			COX-2, IC₅₀: 0.66 μM
COX-2/PI3K-IN-2			COX-2, Ki: 3.02 nM
COX-2/CaV2.2-IN-1			COX-2, IC₅₀: 0.26 μM
Lucidone			COX-2
COX-2-IN-35			COX-2, IC₅₀: 4.37 nM
Andrographidine E			COX-2, IC₅₀: 19 μM
COX-1/2-IN-8		COX-1, IC₅₀: 2.14 ± 0.0 μM	COX-2, IC₅₀: 0.58 ± 0.0 μM
Pifoxime		COX-1	COX-2
COX-2-IN-32			COX-2
WYZ90		COX-1, IC₅₀: 5734 nM	COX-2, IC₅₀: 75 nM
Bromfenac		Human COX-1, IC₅₀: 5.56 nM	Human COX-2, IC₅₀: 7.45 nM
Loxoprofen sodium dihydrate		COX-1, IC₅₀: 6.5 μM (in human whole blood)	COX-2, IC₅₀: 13.5 μM (in human whole blood)
CDK9-IN-41			COX-2, IC₅₀: 775 nM		98.84%
7-Methoxy-4H-chromen-4-one-o-carborane		COX-1, IC₅₀: 3 μM	COX-2, IC₅₀: 1 μM
COX-1-IN-5		COX-1, IC₅₀: 1 nM	COX-2, IC₅₀: >0.1 μM
COX-1-IN-2		COX-1, IC₅₀: 38.76 nM
COX-2-IN-19		COX-1, IC₅₀: 117.8 μM	COX-2, IC₅₀: 1.76 μM
COX-2-IN-52		COX-1, IC₅₀: 15.98 μM	COX-2, IC₅₀: 54 nM
COX-2-IN-66		COX-1, IC₅₀: 32.47 μM	COX-2, IC₅₀: 8.43 μM
COX-2/15-LOX-IN-1		COX-1, IC₅₀: 10.65 μM	COX-2, IC₅₀: 0.075 μM
COX-2-IN-34			COX-2, IC₅₀: 0.42 μM		98.87%
Multitarget AD-IN-3	COX
Santamarine			COX-2		98.85%
Myristinin A			COX-2, IC₅₀: 16.9 μg/mL
Anti-inflammatory agent 78		COX-1	COX-2
COX-2-IN-40			COX-2, IC₅₀: 14.86 μM
COX-2-IN-29		COX-1, IC₅₀: > 10 μM	COX-2, IC₅₀: 0.005 μM
Mefenamic acid-d₄		hCOX-1, IC₅₀: 40 nM	hCOX-2, IC₅₀: 3 nM		98.0%
COX/5-LO-IN-2		COX-1, IC₅₀: 2.95 μM	COX-2, IC₅₀: 1.22 μM
COX-2-IN-42			COX-2
COX-2/5-LOX-IN-6			COX-2, IC₅₀: 2.88 μM
(±)-Aiphanol		COX-1, IC₅₀: 1.9 μM	COX-2, IC₅₀: 9.9 μM
BMP-4 (15-24)			COX-2
COX-2-IN-23		COX-1, IC₅₀: 20.14 μM	COX-2, IC₅₀: 0.28 μM
Anti-inflammatory agent 20			COX-2
CXT29		COX-1, IC₅₀: 722 nM	COX-2, IC₅₀: 13 nM
Zaltoprofen sulfoxide			COX-2, IC₅₀: 45.38 nM
COX-2-IN-20		COX-1, IC₅₀: 19.3 μM	COX-2, IC₅₀: 17.9 nM
α-Amyrin (Standard)			COX-2
Flunixin		COX-1, IC₅₀: 0.55 μM	COX-2, IC₅₀: 3.24 μM
Anti-inflammatory agent 114			COX-2
COX-2-IN-22			COX-2, IC₅₀: 8.6 μM
PPARγ agonist 19		COX-1, IC₅₀: 11.27 μM	COX-2, IC₅₀: 0.05 μM
[10]-Shogaol (Standard)			COX-2, IC₅₀: 7.5 μM
COX-2/NLRP3-IN-1			COX-2, IC₅₀: 1.53 μM
COX-2/Aromatase-IN-2			COX-2
COX-2-IN-43		COX-1, IC₅₀: 0.983 μM	COX-2, IC₅₀: 0.247 μM
MCI			COX-2, IC₅₀: 1.23 μM
COX-2-IN-59		COX-1, IC₅₀: 11.16 μM	COX-2, IC₅₀: 0.052 μM
XO/COX/LOX-IN-1		COX-1, IC₅₀: 12.67 μM	COX-2, IC₅₀: 8.31 μM
Axinelline A		COX-1, IC₅₀: 8.89 μM	COX-2, IC₅₀: 2.22 μM
L 748780		COX-1, IC₅₀: > 100 μM	COX-2, IC₅₀: 0.5 μM
Myristinin B/C			COX-2, IC₅₀: 2.1 μg/mL
DRF-4848			COX-2
COX-2-IN-26		COX-1, IC₅₀: 10.61 μM	COX-2, IC₅₀: 0.067 μM
20(S)-Ginsenoside Rg3 (Standard)			COX-2
Anti-inflammatory agent 56			COX-2
ATP Synthesis-IN-4		COX-1		COX-3
Anti-inflammatory agent 112			COX-2
EGFR/COX-2-IN-2			COX-2, IC₅₀: 50 μM
LY 178002	Cyclooxygenase				99.60%
HDAC6-IN-71			COX-2
Triptolidenol			COX-2
COX-2/5-LOX-IN-7			COX-2, IC₅₀: 3.3 μM
15-LOX-IN-2		COX-1, IC₅₀: 7.510 μM	COX-2, IC₅₀: 0.190 μM
COX-2-IN-61		COX-1, IC₅₀: 43 μM	COX-2, IC₅₀: 22 μM
Dihydroflavokawin B		COX-1, IC₅₀: 1.22 μM	COX-2, IC₅₀: 457 μM
COX-1/2-IN-11		COX-1, : 345 nM	COX-2
Triflusal-d₃		COX-1
COX-2/PI3K-IN-1			COX-2, Ki: 3.24 nM
AS1-6		COX-1, IC₅₀: 12.6 μM	COX-2, IC₅₀: 2.7 μM
Timegadine	COX, IC₅₀: 5 nM (in rabbit platelets) COX, IC₅₀: 20 μM (in rat brain)
2,2'-Biphenol			COX-2
Eltenac		COX-1, IC₅₀: 0.03 μM	COX-2, IC₅₀: 0.03 μM
Multi-kinase-IN-8		COX-1, IC₅₀: 12.6 μM	COX-2, IC₅₀: 0.05 μM
Kaempferol 3-O-(2G-glucosylrutinoside)-7-O-glucoside			COX-2
COX-2/15-LOX-IN-7		COX-1, IC₅₀: 28.081 μM	COX-2, IC₅₀: 0.022 μM
Melafolone			COX-2, IC₅₀: 13.2 μM
Tomoxiprole		COX-1, IC₅₀: 240 nM	COX-2, IC₅₀: 7 nM
COX-2-IN-54			COX-2, IC₅₀: 4.15 μM
Cudraflavone B		COX-1	COX-2
MBL-1			hCOX-2, IC₅₀: 5.77 μM
AChE-IN-82		COX-1, IC₅₀: 60.41 μM	COX-2, IC₅₀: 0.187 μM
Akt/NF-κB/MAPK-IN-1			COX-2
DPAP			COX-2
COX-2-IN-49			COX-2, IC₅₀: 2.671 μM
PYZ18			COX-2, IC₅₀: 7.07 μM
Avicularin (Standard)			COX-2
COX-2-IN-44		COX-1, IC₅₀: 1.14 μM	COX-2, IC₅₀: 0.18 μM
GABAAR/5-HT2AR modulator-1			COX-2
Speranskoside			COX-2, IC₅₀: 2.62 μg/mL
COX-2-IN-24			COX-2, IC₅₀: 0.17 μM
PI3K/AKT-IN-6			COX-2
COX-2/5-LOX-IN-3		COX-1, IC₅₀: 45.73 μM	COX-2, IC₅₀: 5.45 μM
Akt/NF-κB/JNK-IN-1			COX-2
COX-2-IN-57			COX-2, IC₅₀: 0.02 μM
TLR4-IN-2			COX-2
4-Methoxycinnamic acid ethyl ester		COX-1, IC₅₀: 1.12 μM	COX-2, IC₅₀: 0.83 μM		98.72%
RS-57067			COX-2, Ki: 16.9 μM
Triflusal (Standard)		COX-1
Licoflavanone			COX-2
N-(p-Coumaroyl) Serotonin (Standard)			COX-2
NCX 466		COX-1	COX-2
COX-1/2-IN-10		COX-1	COX-2
Indomethacin N-octyl amide		COX-1, IC₅₀: 66 μM	COX-2, IC₅₀: 0.04 μM
N-Caffeoyl serotonin			COX-2, IC₅₀: 42.5 μM
Patrinoside aglucone			COX-2
BF389		COX-1, IC₅₀: 4 μg/mL	COX-2, IC₅₀: 8 μg/mL
Fenoprofen Calcium	COX
COX-1/2-IN-9		COX-1, IC₅₀: 0.031 μM	COX-2, IC₅₀: 0.010 μM
Neosakuranin		COX-1
Balanophonin			COX-2
Multinoside A			COX-2
Tenidap sodium		COX-1	COX-2
4-Desmethyl-2-methyl celecoxib			COX-2, IC₅₀: 0.069 μM
LFS-1107			COX-2
Methosulide		COX-1, IC₅₀: >100 μM	COX-2, IC₅₀: 2.31 μM
ZLJ-6		COX-1, IC₅₀: 0.73 μM	COX-2, IC₅₀: 0.31 μM
Flosulide			COX-2
Thioflosulide			COX-2, IC₅₀: 2.3 nM
S-2474		COX-1, IC₅₀: 27 μM	COX-2, IC₅₀: 11 nM
Saponarin (Standard)			COX-2
SARS-CoV-2 Mpro-IN-41		COX-1, IC₅₀: 46.11 μM	COX-2, IC₅₀: 9.66 μM
Catechin hydrate		COX-1, IC₅₀: 1.4 μM
N1-Acetyl-5-methoxykynuramine hydrochloride			COX-2
Nimesulide-d₅			COX-2, IC₅₀: 0.07-70 μM
COX-2-IN-1			COX-2, IC₅₀: 3.9 μM
COX-2-IN-2			COX-2, IC₅₀: 240 nM		99.53%
Tilmacoxib			Human COX-2, IC₅₀: 85 nM		99.0%
COX/5-LO-IN-1	COX
SC58451			COX-2

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