1. Signaling Pathways
  2. Protein Tyrosine Kinase/RTK
  3. PDGFR
  4. PDGFRα Inhibitors

PDGFRα Inhibitors

PDGFR

PDGFRβ

PDGFRα

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Sorry. There is currently no product that acts on isoform PDGFRα together.

Please try each isoform separately.

PDGFRα Specific Inhibitors
Product Name PDGFRα PDGFRβ PDGFRα Selectivity Purity
Ripretinib
PDGFRA
  Selective Inhibitor 99.46%
Amuvatinib
PDGFRαV561D, IC50: 40 nM
PDGFRαD842V, IC50: 81 nM
  Selective Inhibitor 99.36%
Tyrosine kinase-IN-1
PDGFRα, IC50: 4 nM
  Selective Inhibitor 99.47%
PDGFRα kinase inhibitor 1
PDGFRα, IC50: 132 nM
PDGFRβ, IC50: 6115 nM
Selective Inhibitor
Amuvatinib hydrochloride
PDGFRαV561D, IC50: 40 nM
PDGFRαD842V, IC50: 81 nM
  Selective Inhibitor
Nintedanib
PDGFRα, IC50: 59 nM
PDGFRβ, IC50: 65 nM
Pan Inhibitor 99.97%
Lenvatinib
PDGFRα, IC50: 51 nM
PDGFRβ, IC50: 39 nM
Pan Inhibitor 99.74%
Ilorasertib hydrochloride
PDGFRα, IC50: 11 nM
PDGFRβ, IC50: 13 nM
Pan Inhibitor
Lenvatinib mesylate
PDGFRα, IC50: 51 nM
PDGFRβ, IC50: 39 nM
Pan Inhibitor
Crenolanib
PDGFRα, Kd: 2.1 nM
PDGFRβ, Kd: 3.2 nM
Pan Inhibitor 99.67%
Cediranib
PDGFRα, IC50: 36 nM
PDGFRβ, IC50: 5 nM
Pan Inhibitor 99.58%
Nintedanib esylate
PDGFRα, IC50: 59 nM
PDGFRβ, IC50: 65 nM
Pan Inhibitor 99.95%
CP-673451
PDGFRα, IC50: 10 nM
PDGFRβ, IC50: 1 nM
Pan Inhibitor 99.65%
Dovitinib
PDGFRα, IC50: 27 nM
PDGFRβ, IC50: 210 nM
Pan Inhibitor 97.18%
Telatinib
PDGFRα, IC50: 15 nM
  Pan Inhibitor 99.49%
TAK-593
PDGFRα, IC50: 4.3 nM
PDGFRαV561D, IC50: 1 nM
PDGFRβ, IC50: 13 nM
Pan Inhibitor 99.62%
Cediranib maleate
PDGFRα, IC50: 36 nM
PDGFRβ, IC50: 5 nM
Pan Inhibitor 96.67%
AC710
PDGFRα, Kd: 1.3 nM
PDGFRβ, Kd: 1 nM
Pan Inhibitor 98.03%
Ilorasertib
PDGFRα, IC50: 11 nM
PDGFRβ, IC50: 13 nM
Pan Inhibitor
GZD856
PDGFRα, IC50: 68.6 nM
PDGFRβ, IC50: 136.6 nM
Pan Inhibitor
AC710 Mesylate
PDGFRα, Kd: 1.3 nM
PDGFRβ, Kd: 1 nM
Pan Inhibitor