1. Signaling Pathways
  2. Protein Tyrosine Kinase/RTK
  3. PDGFR
  4. PDGFRβ Inhibitors

PDGFRβ Inhibitors

PDGFR

PDGFRβ

PDGFRα

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Sorry. There is currently no product that acts on isoform PDGFRβ together.

Please try each isoform separately.

PDGFRβ Specific Inhibitors
Product Name PDGFRβ PDGFR PDGFRα PDGFRβ Selectivity Purity
Regorafenib
PDGFRβ, IC50: 22 nM
    Selective Inhibitor 99.96%
Sunitinib
PDGFRβ, IC50: 2 nM
    Selective Inhibitor 99.11%
Sunitinib Malate
PDGFRβ, IC50: 2 nM
    Selective Inhibitor 99.47%
Axitinib
PDGFRβ, IC50: 1.6 nM
    Selective Inhibitor 99.94%
SU 5402
PDGFRβ, IC50: 510 nM
    Selective Inhibitor 99.39%
CP-673451
PDGFRβ, IC50: 1 nM
 
PDGFRα, IC50: 10 nM
Selective Inhibitor 99.65%
Linifanib
PDGFRβ, IC50: 66 nM
    Selective Inhibitor 99.72%
Pazopanib Hydrochloride
PDGFRβ, IC50: 84 nM
    Selective Inhibitor 99.83%
SU14813
PDGFRβ, IC50: 4 nM
    Selective Inhibitor 98.90%
Regorafenib monohydrate
PDGFRβ, IC50: 22 nM
    Selective Inhibitor 99.96%
TG 100801
PDGFRβ, IC50: 13 nM
    Selective Inhibitor 98.60%
Orantinib
PDGFRβ, Ki: 8 nM
    Selective Inhibitor 98.80%
Toceranib phosphate
PDGFRβ, Ki: 5 nM
    Selective Inhibitor 98.43%
Toceranib
PDGFRβ, Ki: 5 nM
    Selective Inhibitor 96.25%
JNJ-10198409
PDGFRβ, IC50: 4.2 nM
 
PDGFRα, IC50: 45 nM
Selective Inhibitor >99.0%
SU14813 maleate
PDGFRβ, IC50: 4 nM
    Selective Inhibitor 99.95%
SU16f
PDGFRβ, IC50: 10 nM
PDGFR2, IC50: 140 nM
PDGFR1, IC50: 2.29 μM
  Selective Inhibitor >99.0%
NVP-ACC789
PDGFR-β, IC50: 1.4 μM
    Selective Inhibitor 99.58%
Tyrphostin AG1433
PDGFRβ, IC50: 5 μM
    Selective Inhibitor 99.20%
AZD2932
PDGFRβ, IC50: 4 nM
    Selective Inhibitor 98.12%
Lenvatinib
PDGFRβ, IC50: 39 nM
 
PDGFRα, IC50: 51 nM
Pan Inhibitor 99.74%
Nintedanib
PDGFRβ, IC50: 65 nM
 
PDGFRα, IC50: 59 nM
Pan Inhibitor 99.97%
PD-089828
PDGFR-β, IC50: 1.76 μM
PDGFR-β, Ki: 2.38 μM
    Pan Inhibitor
Tyrphostin AG1296
PDGFRβ
 
PDGFRα
Pan Inhibitor
Crenolanib
PDGFRβ, Kd: 3.2 nM
 
PDGFRα, Kd: 2.1 nM
Pan Inhibitor 99.67%
Nintedanib esylate
PDGFRβ, IC50: 65 nM
 
PDGFRα, IC50: 59 nM
Pan Inhibitor 99.93%
Cediranib
PDGFRβ, IC50: 5 nM
 
PDGFRα, IC50: 36 nM
Pan Inhibitor 99.58%
Dovitinib
PDGFRβ, IC50: 210 nM
 
PDGFRα, IC50: 27 nM
Pan Inhibitor 97.18%
Regorafenib Hydrochloride
PDGFRβ, IC50: 22 nM
    Pan Inhibitor 99.58%
Dovitinib lactate
PDGFRβ, IC50: 210 nM
 
PDGFRα, IC50: 27 nM
Pan Inhibitor 99.96%
Ilorasertib hydrochloride
PDGFRβ, IC50: 13 nM
 
PDGFRα, IC50: 11 nM
Pan Inhibitor 98.91%
TAK-593
PDGFRβ, IC50: 13 nM
 
PDGFRα, IC50: 4.3 nM
PDGFRαV561D, IC50: 1 nM
Pan Inhibitor 99.62%
Cediranib maleate
PDGFRβ, IC50: 5 nM
 
PDGFRα, IC50: 36 nM
Pan Inhibitor 96.67%
Lenvatinib mesylate
PDGFRβ, IC50: 39 nM
 
PDGFRα, IC50: 51 nM
Pan Inhibitor 98.54%
AC710
PDGFRβ, Kd: 1 nM
 
PDGFRα, Kd: 1.3 nM
Pan Inhibitor 98.03%
PDGFRα kinase inhibitor 1
PDGFRβ, IC50: 6115 nM
 
PDGFRα, IC50: 132 nM
Pan Inhibitor 99.90%
PD-161570
PDGFRβ, IC50: 262 nM
PDGFR, IC50: 310 nM
  Pan Inhibitor
Hypothemycin
PDGFRβ, Ki: 900 nM
 
PDGFRα, Ki: 1.5 μM
Pan Inhibitor
JI-101
PDGFRβ
    default Inhibitor 99.95%