1. Signaling Pathways
  2. Protein Tyrosine Kinase/RTK
  3. PDGFR
  4. PDGFRβ Inhibitors

PDGFRβ Inhibitors

PDGFR

PDGFRβ

PDGFRα

Your Search Returned No Results.

Sorry. There is currently no product that acts on isoform PDGFRβ together.

Please try each isoform separately.

PDGFRβ Specific Inhibitors
Product Name PDGFRβ PDGFR PDGFRα PDGFRβ Selectivity Purity
Regorafenib
PDGFRβ, IC50: 22 nM
    Selective Inhibitor 99.96%
Sunitinib
PDGFRβ, IC50: 2 nM
    Selective Inhibitor 99.66%
SU16f
PDGFRβ, IC50: 10 nM
PDGFR2, IC50: 140 nM
PDGFR1, IC50: 2.29 μM
  Selective Inhibitor >99.0%
Axitinib
PDGFRβ, IC50: 1.6 nM
    Selective Inhibitor 99.94%
SU 5402
PDGFRβ, IC50: 510 nM
    Selective Inhibitor 99.39%
CP-673451
PDGFRβ, IC50: 1 nM
 
PDGFRα, IC50: 10 nM
Selective Inhibitor 99.65%
Sunitinib Malate
PDGFRβ, IC50: 2 nM
    Selective Inhibitor 99.47%
Linifanib
PDGFRβ, IC50: 66 nM
    Selective Inhibitor 99.60%
SU14813
PDGFRβ, IC50: 4 nM
    Selective Inhibitor 98.90%
Pazopanib Hydrochloride
PDGFRβ, IC50: 84 nM
    Selective Inhibitor 99.83%
Toceranib phosphate
PDGFRβ, Ki: 5 nM
    Selective Inhibitor 98.43%
Regorafenib monohydrate
PDGFRβ, IC50: 22 nM
    Selective Inhibitor 99.96%
Toceranib
PDGFRβ, Ki: 5 nM
    Selective Inhibitor 96.25%
SU14813 maleate
PDGFRβ, IC50: 4 nM
    Selective Inhibitor 99.95%
Orantinib
PDGFRβ, Ki: 8 nM
    Selective Inhibitor 98.80%
NVP-ACC789
PDGFR-β, IC50: 1.4 μM
    Selective Inhibitor 99.58%
AZD2932
PDGFRβ, IC50: 4 nM
    Selective Inhibitor 98.12%
JNJ-​10198409
PDGFRβ, IC50: 4.2 nM
 
PDGFRα, IC50: 45 nM
Selective Inhibitor >99.0%
Tyrphostin AG1433
PDGFRβ, IC50: 5 μM
    Selective Inhibitor 99.20%
Sunitinib D10
PDGFRβ, IC50: 2 nM
    Selective Inhibitor
Lenvatinib
PDGFRβ, IC50: 39 nM
 
PDGFRα, IC50: 51 nM
Pan Inhibitor 99.74%
Nintedanib
PDGFRβ, IC50: 65 nM
 
PDGFRα, IC50: 59 nM
Pan Inhibitor 99.97%
Crenolanib
PDGFRβ, Kd: 3.2 nM
 
PDGFRα, Kd: 2.1 nM
Pan Inhibitor 99.67%
Cediranib
PDGFRβ, IC50: 5 nM
 
PDGFRα, IC50: 36 nM
Pan Inhibitor 99.58%
Nintedanib esylate
PDGFRβ, IC50: 65 nM
 
PDGFRα, IC50: 59 nM
Pan Inhibitor 99.95%
Dovitinib
PDGFRβ, IC50: 210 nM
 
PDGFRα, IC50: 27 nM
Pan Inhibitor 97.18%
Regorafenib Hydrochloride
PDGFRβ, IC50: 22 nM
    Pan Inhibitor 99.58%
TAK-593
PDGFRβ, IC50: 13 nM
 
PDGFRα, IC50: 4.3 nM
PDGFRαV561D, IC50: 1 nM
Pan Inhibitor 99.62%
Cediranib maleate
PDGFRβ, IC50: 5 nM
 
PDGFRα, IC50: 36 nM
Pan Inhibitor 96.67%
Ilorasertib hydrochloride
PDGFRβ, IC50: 13 nM
 
PDGFRα, IC50: 11 nM
Pan Inhibitor 98.91%
AC710
PDGFRβ, Kd: 1 nM
 
PDGFRα, Kd: 1.3 nM
Pan Inhibitor 98.03%
PDGFRα kinase inhibitor 1
PDGFRβ, IC50: 6115 nM
 
PDGFRα, IC50: 132 nM
Pan Inhibitor 99.90%
Ilorasertib
PDGFRβ, IC50: 13 nM
 
PDGFRα, IC50: 11 nM
Pan Inhibitor
Lenvatinib mesylate
PDGFRβ, IC50: 39 nM
 
PDGFRα, IC50: 51 nM
Pan Inhibitor
GZD856
PDGFRβ, IC50: 136.6 nM
 
PDGFRα, IC50: 68.6 nM
Pan Inhibitor
AC710 Mesylate
PDGFRβ, Kd: 1 nM
 
PDGFRα, Kd: 1.3 nM
Pan Inhibitor
JI-101
PDGFRβ
    default Inhibitor 99.95%