1. Signaling Pathways
  2. Metabolic Enzyme/Protease
  3. Phospholipase
  4. Phospholipase Inhibitors

Phospholipase Inhibitors

Phospholipase A

PLD

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

Phospholipase Inhibitors & Antagonists
Product Name Phospholipase A PLD Purity
A3373  
PLD1, IC50: 325 nM
PLD2, IC50: 15.15 μM
99.06%
Varespladib
sPLA2, IC50: 9 nM
  99.94%
Bromoenol lactone
PLA2, IC50: 7 μM
  98.41%
1-Naphthaleneacetic acid
PLA2, IC50: 13.16 μM
  99.89%
Pyrrophenone
cPLA2α, IC50: 4.2 nM
  99.76%
VU0155069  
PLD1, IC50: 46 nM
PLD2, IC50: 933 nM
98.04%
Halopemide  
PLD1, IC50: 220 nM
PLD2, IC50: 310 nM
99.65%
OBAA
PLA2, IC50: 70 nM
  99.27%
PACOCF3
PLA2, IC50: 3.8 μM
  ≥98.0%
VU0359595  
PLD1, IC50: 3.7 nM
PLD2, IC50: 6.4 μM
99.65%
sPLA2 inhibitor 1
sPLA2, IC50: 29 nM
  99.47%
Rapanone
PLA2, IC50: 2.6 μM
  99.20%
Alminoprofen
sPLA2
  99.91%
trans-Benzylideneacetone
PLA2
  99.29%
CAY10502
cPLA2α, IC50: 4.3 nM
  ≥99.0%
(S)-Bromoenol lactone
PLA2
  ≥99.0%
VU533  
PLD1, EC50: 0.3 μM
99.71%
CAY10590
sPLA2
  ≥98.0%
(Z)-Oleyloxyethyl phosphorylcholine
sPLA2
 
Lp-PLA2-IN-1
Lp-PLA2
  99.18%
Giripladib
cPLA2α
  99.68%
Varespladib sodium
sPLA2, IC50: 9 nM
  ≥98.0%
BML-280  
PLD2
PLD1
99.64%
1-Naphthaleneacetic acid potassium salt
PLA2, IC50: 13.16 μM
  99.64%
Lp-PLA2-IN-2
Lp-PLA2, IC50: 120 nM
 
YM-26734
sPLA2
 
VI-60
cPLA2
 
Efipladib
cPLA2α, IC50: 0.04 μM
cPLA2α, Ki: 0.067 μM
 
VU0155069 hydrochloride  
PLD1, IC50: 46 nM
SB-435495 hydrochloride
Lp-PLA2, IC50: 0.06 nM
 
Protizinic acid
PLA2, IC50: 210 μM
 
VU 0364739 hydrochloride  
PLD2, IC50: 20 nM
PLD1, IC50: 1500 nM
AX048
cPLA2
 
Lp-PLA2-IN-14
rhLp-PLA2, pIC50: 8.4
 
SB-435495 ditartrate
Lp-PLA2, IC50: 0.06 nM
 
Me-Indoxam
sPLA2
 
SB-435495
Lp-PLA2, IC50: 0.06 nM
  99.80%
FKGK11
PLA2
 
LY 178002
PLA2, IC50: 6.3 μM