1. Signaling Pathways
  2. Metabolic Enzyme/Protease
  3. Phospholipase
  4. Phospholipase Inhibitors

Phospholipase Inhibitors

Phospholipase A

PLD

Phospholipase C

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

Phospholipase Inhibitors, Antagonists, Activators & Substrates
Product Name Phospholipase A PLD Phospholipase C Purity
Ranakinin    
PLC
Varespladib
sPLA2, IC50: 9 nM
    99.74%
Pyrrophenone
cPLA2α, IC50: 4.2 nM
    99.66%
FIPI  
PLD1
PLD2
  98.00%
Bromoenol lactone
PLA2, IC50: 7 μM
    99.59%
1-Naphthaleneacetic acid
PLA2, IC50: 13.16 μM
    99.65%
VU0359595  
PLD1, IC50: 3.7 nM
PLD2, IC50: 6.4 μM
  98.06%
VU0155069  
PLD1, IC50: 46 nM
PLD2, IC50: 933 nM
  98.55%
OBAA
PLA2, IC50: 70 nM
    99.31%
KH064
sPLA2, IC50: 29 nM
    99.84%
SB-435495
Lp-PLA2, IC50: 0.06 nM
    99.71%
OXA(17-33)  
PLD1
 
Varespladib sodium
sPLA2, IC50: 9 nM
    98.83%
Giripladib
cPLA2α
    99.68%
CAY10502
cPLA2α, IC50: 4.3 nM
    ≥99.0%
Rapanone
PLA2, IC50: 2.6 μM
    99.93%
PACOCF3
PLA2, IC50: 3.8 μM
    98.0%
1-Naphthaleneacetic acid potassium salt
PLA2, IC50: 13.16 μM
    99.64%
VU533  
PLD1, EC50: 0.3 μM
  99.84%
N-Palmitoyl-l-leucine
sPLA2
    99.98%
Lp-PLA2-IN-1
Lp-PLA2
    99.30%
Halopemide  
PLD1, IC50: 220 nM
PLD2, IC50: 310 nM
  99.65%
trans-Benzylideneacetone
PLA2
    99.87%
(S)-Bromoenol lactone
PLA2
    99.1%
Alminoprofen
sPLA2
    99.91%
A3373  
PLD1, IC50: 325 nM
PLD2, IC50: 15.15 μM
  99.57%
BML-280  
PLD2
PLD1
  99.64%
Phospholipase C    
PLC
Ochnaflavone
sPLA2, IC50: 3.45 μM
    98.30%
YM-26734
sPLA2
    99.7%
FKGK11
PLA2
    99.9%
LY433771
sPLA2, IC50: 3 nM
    99.8%
(Z)-Oleyloxyethyl phosphorylcholine
sPLA2
    98.0%
Efipladib
cPLA2α, IC50: 0.04 μM
cPLA2α, Ki: 0.067 μM
   
VU 0364739 hydrochloride  
PLD2, IC50: 20 nM
PLD1, IC50: 1500 nM
 
CAY10590
sPLA2
    98.0%
(2E)-OBAA
PLA2, IC50: 70 nM
   
AZD2716
sPLA2
    99.9%
FIPI hydrochloride  
PLD1
PLD2
 
Lp-PLA2-IN-2
Lp-PLA2, IC50: 120 nM
   
VI-60
cPLA2
   
LY256548
PLA2
   
VU0155069 hydrochloride  
PLD1, IC50: 46 nM
 
SB-435495 hydrochloride
Lp-PLA2, IC50: 0.06 nM
   
Protizinic acid
PLA2, IC50: 210 μM
   
PC(O-16:0/18:2(9Z,12Z))
PLA2
   
Parameritannin A-1
PLA2
   
M119    
PLC
AX048
cPLA2
   
BMS-229724
cPLA2
   
WAY-196025
cPLA2α, IC50: 0.01 μM
cPLA2α, Kd: 0.013 μM
   
ML256
Lp-PLA2
   
AGN-190383
PLA2
   
Ro 23-9358
PLA2
   
ASM-IN-2    
PLC, IC50: 0.87 μM
Manoalogue
sPLA2
   
Lp-PLA2-IN-14
rhLp-PLA2, pIC50: 8.4
   
U 84569    
PLC
sPLA2 inhibitor 2
sPLA2, IC50: 0.0475 μM
   
SB-435495 ditartrate
Lp-PLA2, IC50: 0.06 nM
   
LY 178002
PLA2, IC50: 6.3 μM
    99.60%
Me-Indoxam
sPLA2
   
SHP1-IN-2    
PLC
PLA2-IN-1
PLA2, IC50: 1 nM
   
Cinatrin C2
PLA2, IC50: 800 μM
   
BAPTA tetracesium    
PLC
Cinatrin C3
PLA2, IC50: 70 μM
   
Cinatrin C1
PLA2
   
Darapladib analog-1
Lp-PLA2