1143578-94-2
Chemical Structure
FAAH-IN-6
- CAS No.: 1143578-94-2
- Formula:C19H17F2N7O
- Molecular Weight:397.38
IUPAC Name: 4-(4-(3,4-difluorophenyl)pyrimidin-2-yl)-N-(pyridazin-3-yl)piperazine-1-carboxamide
InChIKey: JCWVFSJNIBAGQN-UHFFFAOYSA-N
SMILES: O=C(N1CCN(C2=NC=CC(C3=CC=C(F)C(F)=C3)=N2)CC1)NC4=NN=CC=C4
Biological Activity: FAAH-IN-6 (compound 21d) is a potent, orally active and cross the blood-brain barrier fatty acid amide hydrolase (FAAH) inhibitor with IC50s of 0.72, 0.28 nM for hFAAH, rFAAH, respectively. FAAH-IN-6 shows dose-dependent analgesic efficacy in animal models of both neuropathic and inflammatory pain[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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FAAH-IN-6 | 99.70% | FAAH-IN-6 (compound 21d) is a potent, orally active and cross the blood-brain barrier fatty acid amide hydrolase (FAAH) inhibitor with IC50s of 0.72, 0.28 nM for hFAAH, rFAAH, respectively. FAAH-IN-6 shows dose-dependent analgesic efficacy in animal models of both neuropathic and inflammatory pain. | ||||||||||||||||||||
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Keywords
