1221964-37-9
1221964-37-9
Chemical Structure
PS423
- CAS No.: 1221964-37-9
- Formula:C25H23F3O9
- Molecular Weight:524.44
IUPAC Name: bis(acetoxymethyl) 2-(3-oxo-1-phenyl-3-(4-(trifluoromethyl)phenyl)propyl)malonate
InChIKey: KNHNCABHIAKMBD-UHFFFAOYSA-N
SMILES: O=C(OCOC(C)=O)C(C(C1=CC=CC=C1)CC(C2=CC=C(C(F)(F)F)C=C2)=O)C(OCOC(C)=O)=O
Biological Activity: PS423 is a prodrug of PS210, acting as a substrate-selective inhibitor of PDK1, inhibiting the phosphorylation and activation of S6K. PS210 is a potent and selective PDK1 activator targeting the PIF binding pocket of PDK1[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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PS423 | 99.38% | PS423 is a prodrug of PS210, acting as a substrate-selective inhibitor of PDK1, inhibiting the phosphorylation and activation of S6K. PS210 is a potent and selective PDK1 activator targeting the PIF binding pocket of PDK1. | ||||||||||||||||||||
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References
Keywords
