2309762-30-7
Chemical Structure
Elacestrant S enantiomer dihydrochloride
Synonym(s): RAD1901 S enantiomer dihydrochloride
- CAS No.: 2309762-30-7
- Formula:C30H40Cl2N2O2
- Molecular Weight:531.56
IUPAC Name: (S)-6-(2-(ethyl(4-(2-(ethylamino)ethyl)benzyl)amino)-4-methoxyphenyl)-5,6,7,8-tetrahydronaphthalen-2-ol dihydrochloride
InChIKey: XGFHYCAZOCBCRQ-ROPHLPQBSA-N
SMILES: OC1=CC=C2C[C@@H](C3=CC=C(OC)C=C3N(CC)CC4=CC=C(CCNCC)C=C4)CCC2=C1.[H]Cl.[H]Cl
Biological Activity: Elacestrant S enantiomer dihydrochloride (RAD1901 S enantiomer dihydrochloride) is an low activity enantiomer of elacestrant dihydrochloride. Elacestrant (RAD1901) dihydrochloride is a selective and orally available estrogen receptor (ERR) degrader with IC50 values of 48 and 870 nM for ERα and ERβ, respectively.
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Elacestrant S enantiomer dihydrochloride | Elacestrant S enantiomer dihydrochloride (RAD1901 S enantiomer dihydrochloride) is an low activity enantiomer of elacestrant dihydrochloride. Elacestrant (RAD1901) dihydrochloride is a selective and orally available estrogen receptor (ERR) degrader with IC50 values of 48 and 870 nM for ERα and ERβ, respectively. | |||||||||||||||||||||
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