3036054-38-0
3036054-38-0
Chemical Structure
CARM1-IN-5
- CAS No.: 3036054-38-0
- Formula:C22H26ClN3O2S
- Molecular Weight:431.98
InChIKey: UMKLFWMQTDMELK-SFHVURJKSA-N
SMILES: CN(CC1=CC=CC=C1OCC2=CC(Cl)=C(C=C2)C3=NC=CS3)C[C@H](CNC)O
Biological Activity: CARM1-IN-5 (Compound 17e) is a potent and selective inhibitor of CARM1 (IC50= 2 nM). CARM1-IN-5 effectively prevents CARM1 from methylating substrate proteins by directly interacting with CARM1. CARM1-IN-5 exhibits significant antiproliferative effects on melanoma cell lines[1].
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CARM1-IN-5 | CARM1-IN-5 (Compound 17e) is a potent and selective inhibitor of CARM1 (IC50= 2 nM). CARM1-IN-5 effectively prevents CARM1 from methylating substrate proteins by directly interacting with CARM1. CARM1-IN-5 exhibits significant antiproliferative effects on melanoma cell lines. | |||||||||||||||||||||
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References
Keywords
