3037016-67-1
3037016-67-1
Chemical Structure
Keap1-Nrf2-IN-6
- CAS No.: 3037016-67-1
- Formula:C30H34N4O8S
- Molecular Weight:610.68
IUPAC Name: (R)-7-chloro-2-((1r,4R)-4-(3-methoxyazetidin-1-yl)cyclohexyl)-2,4-dimethyl-N-((6-methyl-4-(methylthio)-2-oxo-1,2-dihydropyridin-3-yl)methyl)benzo[d][1,3]dioxole-5-carboxamide
InChIKey: RNGXYARCEQWNBD-SDHSZQHLSA-N
SMILES: O=C1N[C@H](CSCC2=C(C(OC[C@H]1NC([C@@H]3CCCN3C(C)=O)=O)=O)C=CC=C2C4=CC=C(C=C4)C(O)=O)C(N(C)C)=O
Biological Activity: Keap1-Nrf2-IN-6 (compound 64) is a potent and selective Keap1-Nrf2 PPI (Keap1-Nrf2 protein−protein interaction) inhibitor with an IC50 of 41 nM, Kd of 68 nM[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
|
|
Keap1-Nrf2-IN-6 | Keap1-Nrf2-IN-6 (compound 64) is a potent and selective Keap1-Nrf2 PPI (Keap1-Nrf2 protein−protein interaction) inhibitor with an IC50 of 41 nM, Kd of 68 nM. | |||||||||||||||||||||
|
loading...
/
|
|||||||||||||||||||||||
References
Keywords
