870281-82-6
870281-82-6
Chemical Structure
Idelalisib
Synonym(s): CAL-101; GS-1101
- CAS No.: 870281-82-6
- Formula:C22H18FN7O
- Molecular Weight:415.42
IUPAC Name: (S)-2-(1-((9H-purin-6-yl)amino)propyl)-5-fluoro-3-phenylquinazolin-4(3H)-one
InChIKey: IFSDAJWBUCMOAH-HNNXBMFYSA-N
SMILES: O=C1N(C2=CC=CC=C2)C([C@@H](NC3=C4N=CNC4=NC=N3)CC)=NC5=C1C(F)=CC=C5
Biological Activity: Idelalisib (CAL-101; GS-1101) is a highly selective and orally bioavailable p110δ inhibitor with an IC50 of 2.5 nM, showing 40- to 300-fold selectivity for p110δ over other PI3K class I enzymes.
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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Idelalisib | 99.94% | Idelalisib (CAL-101; GS-1101) is a highly selective and orally bioavailable p110δ inhibitor with an IC50 of 2.5 nM, showing 40- to 300-fold selectivity for p110δ over other PI3K class I enzymes. | ||||||||||||||||||||
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Idelalisib (Standard) | ≥98% | Idelalisib (Standard) is the analytical standard of Idelalisib. This product is intended for research and analytical applications. Idelalisib (CAL-101; GS-1101) is a highly selective and orally bioavailable p110δ inhibitor with an IC50 of 2.5 nM, showing 40- to 300-fold selectivity for p110δ over other PI3K class I enzymes. | ||||||||||||||||||||
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Idelalisib-d5 | 98.35% | Idelalisib-d5 is a deuterium labeled Idelalisib. Idelalisib is a highly selective and orally bioavailable p110δ inhibitor. | ||||||||||||||||||||
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