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Cat. No.: HY-129224

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XS018661

XS018661 is a dual inhibitor of the YEATS domains of ENL and its paralog AF9 with IC₅₀ values of 1.6 and 3 μM as well as K_d values of 754 nM and 523 nM, respectively.

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CAS No.: 878415-59-9
Formule: C₂₂H₂₄N₄O₃
Masse moléculaire:392.46

Stockage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (264 KB)

XS018661 Chemical Structure

CAS No.: 878415-59-9

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Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Activité biologique

Description

XS018661 is a dual inhibitor of the YEATS domains of ENL and its paralog AF9 with IC₅₀ values of 1.6 and 3 μM as well as K_d values of 754 nM and 523 nM, respectively^[1].

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Chemical Information

CAS No. 878415-59-9
Masse moléculaire 392.46
Formule C₂₂H₂₄N₄O₃
SMILES

O=C(OC)C1=CC=C(C=C1)C(=O)NC=2C=CC=3N=C(NC3C2)CN4CCCCC4
Livraison

Room temperature in continental US; may vary elsewhere.
Stockage

Please store the product under the recommended conditions in the Certificate of Analysis.

Pureté et documentation

Select Batch:

Pureté: 99.98%

Assay: 99.98%

ee.: 99.98%

Fiche technique (264 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Instruction de manipulation (2659 KB)

Références

[1]. Christott T, et al., Discovery of a Selective Inhibitor for the YEATS Domains of ENL/AF9. SLAS Discov. 2019 Feb;24(2):133-141. [Content Brief]

Calculators

Calculateur de molarité

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass Mass

Concentration Concentration

Volume Volume

Molecular Weight Molecular Weight

Calculateur de dilution

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

Concentration _(start) Concentration _(start)

Volume _(start) Volume _(start)

Concentration _(final) Concentration _(final)

Volume _(final) Volume _(final)

Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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100 mg

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XS018661

Voir tous les produits spécifiques à Isoform Epigenetic Reader Domain

Activité biologique

Chemical Information

Pureté et documentation

Références

Calculators

Help & FAQs

XS018661 Related Classifications

HY-129224 Related Classifications