VPC-3033

VPC-3033 is an androgen receptor antagonist. VPC-3033 has a strong androgen DHT replacement potency (IC50: 0.625-2.5 μM), can effectively inhibit androgen receptor transcriptional activity (IC50=0.3 μM), and has a strong androgen receptor degradation ability. In addition, VPC-3033 exhibits significant anti-androgen receptor activity against prostate cancer cells resistant to Enzalutamide (HY-70002).

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  • No. CAS: 110763-24-1
  • Fòrmula: C21H14O2
  • Peso molecular:298.33
  • Almacenamiento:

    Please store the product under the recommended conditions in the Certificate of Analysis.

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