CTR/AMYR agonist-2
CTR/AMYR agonist-2 is a fused heterocyclic amide/sulfonamide compound, as well as a calcitonin G protein-coupled receptor (CGRP Receptor) / amylin receptor agonist. CTR/AMYR agonist-2 shows potential for application in research related to diseases such as obesity and type 2 diabetes.
商品は「研究用試薬」です。人や動物の医療用・臨床診断用・食品用の製品ではありません。
研究用途以外に使用した場合、当社は一切の責任を負いかねます。
- 分子式: C36H35F2N7O6
- 分子量:699.70
-
保管条件:
Please store the product under the recommended conditions in the Certificate of Analysis.
生物活性
製品説明
体外実験
CTR/AMYR agonist-2 (Example 117) exhibits a geometric mean EC50 of 1.89 nM and an asymptotic maximum response of 128% in the HTRF‑cAMP agonism functional assay using CHO cells expressing human calcitonin receptor[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
化学情報
-
分子量 699.70
-
分子式 C36H35F2N7O6
-
SMILES
O[C@@H](C1)[C@@H](NC(C2=COC(C3=C(C4=NN=C(CN(C)C)O4)C(CCC5=CC=C(F)C=C5)=NC(O[C@H](C)[C@@H](C)N6)=C3C6=O)=N2)=O)C7=C1C=C(F)C=C7
-
輸送条件
Room temperature in continental US; may vary elsewhere.
-
保管条件
Please store the product under the recommended conditions in the Certificate of Analysis.
純度とドキュメンテーション
参考文献
Calculators
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)