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Cat. No.: HY-129224

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XS018661

XS018661 is a dual inhibitor of the YEATS domains of ENL and its paralog AF9 with IC₅₀ values of 1.6 and 3 μM as well as K_d values of 754 nM and 523 nM, respectively.

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CAS No.: 878415-59-9
화학식: C₂₂H₂₄N₄O₃
분자량:392.46

보관:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (264 KB)

XS018661 Chemical Structure

CAS No.: 878415-59-9

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Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity

제품 설명

XS018661 is a dual inhibitor of the YEATS domains of ENL and its paralog AF9 with IC₅₀ values of 1.6 and 3 μM as well as K_d values of 754 nM and 523 nM, respectively^[1].

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Chemical Information

CAS No. 878415-59-9
분자량 392.46
화학식 C₂₂H₂₄N₄O₃
SMILES

O=C(OC)C1=CC=C(C=C1)C(=O)NC=2C=CC=3N=C(NC3C2)CN4CCCCC4
선적

Room temperature in continental US; may vary elsewhere.
보관

Please store the product under the recommended conditions in the Certificate of Analysis.

순도&문서

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (264 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

References

[1]. Christott T, et al., Discovery of a Selective Inhibitor for the YEATS Domains of ENL/AF9. SLAS Discov. 2019 Feb;24(2):133-141. [Content Brief]

Calculators

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Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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Concentration Concentration

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Molecular Weight Molecular Weight

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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100 mg

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Chemical Information
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XS018661

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Biological Activity

Chemical Information

순도&문서

References

Calculators

Help & FAQs

XS018661 Related Classifications

HY-129224 Related Classifications