1 Result for "

Crinecerfont (Standard)

" in MedChemExpress (MCE) Product Catalog:
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1 Results for "Crinecerfont (Standard)" in MCE Product Catalog:

Cat. No.: HY-106203R
CAS No.: 752253-39-7
Synonyms: SSR-125543 (Standard)
Research Areas:  

Metabolic Disease

Crinecerfont (Standard) is the analytical standard of Crinecerfont (HY-106203). This product is intended for research and analytical applications. Crinecerfont (SSR-125543) is an orally effective corticotropin-releasing factor receptor type-1 (CRF1 receptor) antagonist. Crinecerfont blocks CRF1 receptor signaling to reduce adrenocorticotropic hormone secretion. Crinecerfont improves hypothalamic-pituitary-adrenal axis negative feedback sensitivity in chronically stressed mice. Crinecerfont can be used for the research of chronic stress conditions and classic congenital adrenal hyperplasia due to 21-hydroxylase deficiency. Crinecerfont is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.
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