1 Result for "

ERβ agonist1

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "ERβ agonist1" in MCE Product Catalog:

Cat. No.: HY-173474
CAS No.: 2412715-30-9
Research Areas:  

Cancer

ERβ agonist-1 (Compound 8) is a dual-active selective ERβ agonist (EC50: 46.8 nM) and AR antagonist (IC50: 1555 nM). ERβ agonist-1 activates ERβ signaling by binding to ERβ and inhibits AR activity. ERβ agonist-1 retains selective ERβ agonist activity in mouse models and can be used to study prostate cancer .
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