4 Results for "

PROTAC CB1R Degrader-1

" in MedChemExpress (MCE) Product Catalog:
Products (4)

4 Results for "PROTAC CB1R Degrader-1" in MCE Product Catalog:

Cat. No.: HY-178176
Research Areas:  

Cancer

PROTAC CB1R Degrader-1 is a potent and selective CB1R PROTAC degrader that exploits the ubiquitin-proteasome system (UPS) achieving a DC50 of 3.37 μM in MCF-7 cells and showing no impact on CB2R. PROTAC CB1R Degrader-1 reduces CB1R-associated downstream signaling (p-AKT, p-ERK, BCL2, and MCM5), thereby inhibiting breast cancer cell proliferation and inducing apoptosis. PROTAC CB1R Degrader-1 can be used for breast cancer research .
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Cat. No.: HY-178198
CAS No.: 87156-42-1
Target:  

PROTAC Linkers

Research Areas:  

Cancer

2-[4-(Aminomethyl)triazol-1-yl]ethanamine is a PROTAC Linker. 2-[4-(Aminomethyl)triazol-1-yl]ethanamine can be used to synthesize PROTAC CB1R Degrader-1 (HY-178176) .
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Cat. No.: HY-134497
CAS No.: 162758-35-2
Synonyms: Rimonabat acomplia
Rimonabant carboxylic acid is a Ligand for Target Protein for PROTAC. Rimonabant carboxylic acid can be used to synthesize PROTAC CB1R Degrader-1 (HY-178176) .
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Cat. No.: HY-178197
Research Areas:  

Cancer

E3 Ligase Ligand-linker Conjugate 210 is an E3 ligase ligand-linker conjugate. E3 Ligase Ligand-linker Conjugate 210 can be used to synthesize PROTAC CB1R Degrader-1 (HY-178176) .
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