42 Results for "

adrenoreceptor

" in MedChemExpress (MCE) Product Catalog:
Products (42)

42 Results for "adrenoreceptor" in MCE Product Catalog:

2
2 Cited Publications
Cat. No.: HY-129041
CAS No.: 81262-93-3
Purity:  99.88%
Synonyms: OPC 2009 hydrochloride hemihydrate
Target:  

Adrenergic Receptor

Research Areas:  

Infection Inflammation/Immunology

Procaterol hydrochloride hemihydrate is an orally active β2 adrenoreceptor agonist. Procaterol hydrochloride hemihydrate can be used for the research of asthma .
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2
2 Cited Publications
Cat. No.: HY-100704
CAS No.: 62929-91-3
Procaterol hydrochloride is a selective intermediate-acting β2 adrenoreceptor agonist with an EC50 of 12.9 μM . Procaterol hydrochloride can inhibit inflammation both in vivo and in vitro .
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1
1 Cited Publications
Cat. No.: HY-105124A
CAS No.: 60398-91-6
Purity:  98.03%
Synonyms: Ro 3-4787 hydrochloride
Target:  

Adrenergic Receptor

Bufuralol (Ro 3-4787) hydrochloride is a potent non-selective, orally active β-adrenoreceptor antagonist with partial agonist activity. Bufuralol hydrochloride is a CYP2D6 probe substrate .
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1
1 Cited Publications
Cat. No.: HY-105124
CAS No.: 54340-62-4
Purity:  99.17%
Synonyms: Ro 3-4787
Target:  

Adrenergic Receptor

Bufuralol (Ro 3-4787) is a potent non-selective, orally active β-adrenoreceptor antagonist with partial agonist activity. Bufuralol hydrochloride is a CYP2D6 probe substrate .
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1
1 Cited Publications
Cat. No.: HY-10564
CAS No.: 135159-51-2
Purity:  99.09%
Synonyms: MCI-9042
Target:  

5-HT Receptor

Research Areas:  

Cardiovascular Disease

Sarpogrelate hydrochloride (MCI-9042) is a selective 5-HT2R antagonist, with pKis of 8.52, 6.57, and 7.43 for 5-HT2A, 5-HT2B, and 5-HT2C receptors, respectively. Sarpogrelate hydrochloride displays selectivity over 5-HT1, 5-HT3, 5-HT4, α1-, α2- and β-adrenoreceptor, histamine H1, H2 and muscarinic M3 receptors. Sarpogrelate hydrochloride can be used for the research of vascular disease associated with thrombosis .
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1
1 Cited Publications
Cat. No.: HY-P81085
Synonyms: Beta 2-adrenergic receptor; beta 2 Adrenergic Receptor; ADRB2R; ADRBR; ADRB2_HUMAN; Adrenergic beta 2 receptor surface; B2AR; BAR; Beta 2 adrenoreceptor; BETA2AR; Catecholamine receptor; beta2-adrenergic receptor. β2-adrenergic receptor;

Host:  

Rabbit

Application:  

WB

Reactivity:  

Human, Mouse, Rat

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Cat. No.: HY-B0716
CAS No.: 34661-75-1
Urapidil is an α1 adrenoreceptor antagonist and a 5-HT1A receptor agonist that can cross the blood-brain barrier .
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Cat. No.: HY-108300
CAS No.: 16777-42-7
Purity:  99.92%
Target:  

Adrenergic Receptor

Research Areas:  

Cardiovascular Disease

Oxyfedrine hydrochloride, a vasodilator, is an orally active β-adrenoreceptor agonist. Oxyfedrine decreases the tonicity of coronary vessels. Oxyfedrine hydrochloride can be used in the research of cardiovascular disease .
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Cat. No.: HY-W153159
CAS No.: 13062-76-5
N-Methyltyramine hydrochloride is an orally active α2-adrenoreceptor antagonist with an IC50 value of 5.53 μM against rat targets. N-Methyltyramine hydrochloride blocks α2-adrenoreceptors, while inhibiting lipolysis, hyperactivity responses and small intestinal peristalsis in mice. N-Methyltyramine hydrochloride promotes gastrin release and pancreatic juice secretion, upregulates appetite, blood pressure, myocardial contraction frequency and contraction intensity, and increases renal blood flow, renal vascular resistance and mean peripheral arterial resistance. N-Methyltyramine hydrochloride relaxes mouse small intestinal smooth muscle and undergoes biotransformation in vivo to produce adrenaline. N-Methyltyramine hydrochloride can be used in studies related to gastrointestinal diseases .
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Cat. No.: HY-17498A
CAS No.: 93379-54-5
Target:  

Adrenergic Receptor

Research Areas:  

Cardiovascular Disease

(S)-Atenolol is a potent beta-adrenoreceptor blocker. (S)-Atenolol has the potential for the research of cardiovascular disorder .
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Cat. No.: HY-112070
CAS No.: 15687-41-9
Target:  

Adrenergic Receptor

Research Areas:  

Cardiovascular Disease

Oxyfedrine, a vasodilator, is an orally active β-adrenoreceptor agonist. Oxyfedrine decreases the tonicity of coronary vessels. Oxyfedrine can be used in the research of cardiovascular disease .
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Cat. No.: HY-B0716S2
CAS No.: 1795122-12-1
Urapidil-d4 is the deuterium labeled Urapidil . Urapidil is an α1 adrenoreceptor antagonist and a 5-HT1A receptor agonist .
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Cat. No.: HY-P5881
Target:  

PKC

Research Areas:  

Cardiovascular Disease

PKCα (C2-4) inhibitor peptide is a PKCα specific inhibitor peptide that blocks the inhibition of IKr by the α1A adrenoreceptor agonist A-61603 (HY-101366) .
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Cat. No.: HY-W153897
CAS No.: 370-98-9
N-Methyltyramine is an orally active α2-adrenoreceptor antagonist with an IC50 value of 5.53 μM against rat targets. N-Methyltyramine blocks α2-adrenoreceptors, while inhibiting lipolysis, hyperactivity responses and small intestinal peristalsis in mice. N-Methyltyramine promotes gastrin release and pancreatic juice secretion, upregulates appetite, blood pressure, myocardial contraction frequency and contraction intensity, and increases renal blood flow, renal vascular resistance and mean peripheral arterial resistance. N-Methyltyramine relaxes mouse small intestinal smooth muscle and undergoes biotransformation in vivo to produce adrenaline. N-Methyltyramine can be used in studies related to gastrointestinal diseases .
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Cat. No.: HY-109130
CAS No.: 1799809-36-1
Synonyms: BAY 1193397
Target:  

Adrenergic Receptor

Research Areas:  

Metabolic Disease

Fadaltran (BAY 1193397) is an orally active α2C-adrenoreceptor antagonist. Fadaltran can be used for the study of diabetic foot ulcers .
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Cat. No.: HY-B0716R
CAS No.: 34661-75-1
Urapidil (Standard) is the analytical standard of Urapidil. This product is intended for research and analytical applications. Urapidil is an α1 adrenoreceptor antagonist and a 5-HT1A receptor agonist that can cross the blood-brain barrier .
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Cat. No.: HY-10564R
CAS No.: 135159-51-2
Synonyms: MCI-9042 (Standard)
Research Areas:  

Cardiovascular Disease

Sarpogrelate (hydrochloride) (Standard) is the analytical standard of Sarpogrelate (hydrochloride). This product is intended for research and analytical applications. Sarpogrelate hydrochloride (MCI-9042) is a selective 5-HT2R antagonist, with pKis of 8.52, 6.57, and 7.43 for 5-HT2A, 5-HT2B, and 5-HT2C receptors, respectively. Sarpogrelate hydrochloride displays selectivity over 5-HT1, 5-HT3, 5-HT4, α1-, α2- and β-adrenoreceptor, histamine H1, H2 and muscarinic M3 receptors. Sarpogrelate hydrochloride can be used for the research of vascular disease associated with thrombosis .
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Cat. No.: HY-111206
CAS No.: 883724-08-1
Target:  

Adrenergic Receptor

Research Areas:  

Inflammation/Immunology

β3-AR agonist 3 is a potent beta-3 adrenoreceptor agonist. β3-AR agonist 3 has the potential for prostatitis research .
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Cat. No.: HY-147299
CAS No.: 177843-85-5
Synonyms: PGE-6201204
Target:  

Adrenergic Receptor

Research Areas:  

Cardiovascular Disease

Povafonidine (PGE-6201204) is a potent α2 adrenoreceptor agonist. Povafonidine can constrict blood vessels and reduce mucosal congestion. Povafonidine can be used for nasal congestion research .
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Cat. No.: HY-128510
CAS No.: 18866-78-9
Target:  

Adrenergic Receptor

Research Areas:  

Cardiovascular Disease

Colterol is the agonist for adrenergic receptor, and exhibits good affinity to β1-adrenoreceptor (heart) and β2-adrenoreceptor (lung) with IC50 of 645 nM and 147 nM. Colterol exhibits potential as a bronchodilator .
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