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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
37 Results for "
cannabinoid-CB1
" in MedChemExpress (MCE) Product Catalog:
Products (37)
37 Results for "cannabinoid-CB1" in MCE Product Catalog:
7
7 Publications Verification
Synonyms: 3β-Hydroxy-5-pregnen-20-one
7
7 Publications Verification
Synonyms: 3β-Hydroxy-5-pregnen-20-one monosulfate
Category:
7
7 Publications Verification
Synonyms: 3β-Hydroxy-5-pregnen-20-one monosulfate sodium
Category:
2
Target:
Research Areas:
Arachidonylcyclopropylamide (ACPA) is a potent and selective CB1 receptors agonist. Arachidonylcyclopropylamide inhibits forskolin-stimulated cAMP production in CHO cells transfected with human cannabinoid CB1 receptors (IC50=2 nM) [1].
1
Category:
other families Other Phenylpropanoids Phenylpropanoids Plants Disease Research Fields Inflammation/Immunology
Target:
1
1 Cited Publications
Synonyms: SLV319; BMS-646256
Target:
Research Areas:
Ibipinabant (SLV319) is a potent, selective and orally active antagonist of cannabinoid CB1 receptor, with a Ki of 7.8 nM. Ibipinabant shows more than 1000-fold selectivity for CB1 over CB2 (Ki=7943 nM). Ibipinabant can be used for the research of obesity and diabetic [1] .
1
1 Cited Publications
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Research Areas:
AZD1940 is an orally active, high affinity cannabinoid CB1/CB2 receptor agonist with pKi values of 7.93 and 9.06 for human CB1R and CB2R, respectively. AZD1940 shows a robust analgesia action [1] .
1
1 Cited Publications
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Research Areas:
NESS 0327 is a cannabinoid antagonist with high selectivity for the cannabinoid CB1 receptor. NESS 0327 is more than 60,000-fold selective for the CB1 receptor [1].
1
1 Cited Publications
Target:
Research Areas:
LH-21 is a potent in vivo neutral cannabinoid CB1 receptor antagonist. LH-21 reduces food intake and body weight gain in obese Zucker rats.
, and displays efficacy as a feeding inhibitor [1].
Target:
Research Areas:
Bay 59-3074 is a selective cannabinoid CB1/CB2 receptor partial agonist with Ki values of 48.3 and 45.5 nM at human CB1 and CB2 receptors, respectively. Bay 59-3074 has analgesic properties [1].
Synonyms: (S)-MRI-1867
Target:
Research Areas:
Zevaquenabant ((S)-MRI-1867) is a peripherally restricted, orally bioavailable dual cannabinoid CB1 receptor and inducible NOS antagonist. Zevaquenabant ameliorates obesity-induced chronic kidney disease (CKD) [1].
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Target:
Cat. No.: HY-124089
CAS No.: 109001-03-8
Target:
Research Areas:
Eicosapentaenoyl ethanolamide, an omega-3 fatty acid, is one of N-acylethanolamines (NAEs). Eicosapentaenoyl ethanolamide is cannabinoid CB1/CB2 receptor agonist. Eicosapentaenoyl ethanolamide acts as a metabolic signal. Eicosapentaenoyl ethanolamide inhibits dietary restriction (DR)-induced lifespan extension in wild type animals and suppresses lifespan extension in a TOR pathway mutant [1] .
Cat. No.: HY-B0151S2
CAS No.: 61574-54-7
Synonyms: 3β-Hydroxy-5-pregnen-20-one-d4-1
Cat. No.: HY-110014
CAS No.: 222723-55-9
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Research Areas:
Noladin ether is a potent and selective agonist of cannabinoid CB1 receptor, with a Ki of 21.2 nM. Noladin ether can cause hypothermia, intestinal immobility, and mild antinociception [1].
Cat. No.: HY-W127407
CAS No.: 201738-25-2
Cat. No.: HY-110189S1
CAS No.: 1485492-21-4
Synonyms: 3β-Hydroxy-5-pregnen-20-one monosulfate-d4 sodium
Cat. No.: HY-128040
CAS No.: 443129-35-9
Research Areas:
Virodhamine (hydrochloride) is a cannabinoid CB1 receptor partial agonist and cannabinoid CB2 receptor full agonist [1].
Cat. No.: HY-133533
CAS No.: 1883545-42-3
Target:
Research Areas:
O-2050 is a high affinity cannabinoid CB1 receptor antagonist with a Ki of 2.5 nM. O-2050 inhibits cannabinoid CB2 receptor (Ki=0.2 nM). O-2050 can cause locomotor stimulation in mice [1].
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Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
