1. GPCR/G Protein
    Neuronal Signaling
  2. mGluR
  3. LY2794193

LY2794193 

Cat. No.: HY-119243 Purity: 99.88%
Handling Instructions

LY2794193 is a highly potent and selective mGlu3 receptor agonist (hmGlu3 Ki=0.927 nM,EC50=0.47 nM; hmGlu2 Ki=412 nM,EC50=47.5 nM).

For research use only. We do not sell to patients.

LY2794193 Chemical Structure

LY2794193 Chemical Structure

CAS No. : 2173037-97-1

Size Price Stock Quantity
5 mg USD 550 In-stock
Estimated Time of Arrival: December 31
10 mg USD 850 In-stock
Estimated Time of Arrival: December 31
50 mg USD 2850 In-stock
Estimated Time of Arrival: December 31
100 mg USD 3950 In-stock
Estimated Time of Arrival: December 31
200 mg   Get quote  
500 mg   Get quote  

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Customer Review

Based on 1 publication(s) in Google Scholar

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Description

LY2794193 is a highly potent and selective mGlu3 receptor agonist (hmGlu3 Ki=0.927 nM,EC50=0.47 nM; hmGlu2 Ki=412 nM,EC50=47.5 nM)[1].

IC50 & Target[1]

mGluR3

0.47 nM (EC50)

mGluR3

0.927 nM (Ki)

mGluR2

47.5 (EC50)

mGluR2

412 (Ki)

Molecular Weight

334.32

Formula

C₁₆H₁₈N₂O₆

CAS No.

2173037-97-1

SMILES

O=C([[email protected]@]1(N)[[email protected]]2([H])[[email protected]@H](C(O)=O)[[email protected]]2([H])[[email protected]@H](NC(C3=CC=CC(OC)=C3)=O)C1)O

Shipping

Room temperature in continental US; may vary elsewhere

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
Solvent & Solubility
In Vitro: 

H2O : 2 mg/mL (5.98 mM; ultrasonic and adjust pH to 14 with NaOH)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.9911 mL 14.9557 mL 29.9115 mL
5 mM 0.5982 mL 2.9911 mL 5.9823 mL
10 mM --- --- ---
*Please refer to the solubility information to select the appropriate solvent.
References
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Product Name:
LY2794193
Cat. No.:
HY-119243
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