Leukotriene Receptor Inhibitors

LTB₄

LTC₄

LTD₄/CysLT₁

LTE₄

CysLT₂

CysLT₁

Leukotriene Receptor Inhibitors, Agonists & Antagonists

Product Name	LTB₄	LTC₄	LTD₄/CysLT₁	LTE₄	CysLT₂	CysLT₁	Purity
MK-571 sodium			LTD₄, Ki: 0.22±0.15 nM (In guinea pig lung) LTD₄, Ki: 2.1±1.8 nM (In human lung) LTD₄, pA2: 10.5	LTE₄, pA2: 10.4			99.24%
Montelukast sodium						CysLT₁	99.52%
Zafirlukast			LTD₄				99.90%
LTB4 antagonist 1	LTB₄
CP-195543	LTB₄
LTB4 antagonist 2	LTB₄, IC₅₀: 439 nM
LY255283	LTB₄, IC₅₀: ~100 nM (LTB₄ binds to guinea pig lung membranes)						98.73%
CP-105696	LTB₄, IC₅₀: 8.42±0.26 nM						99.66%
Gemilukast					CysLT₂, IC₅₀: 25 nM (in human)	CysLT₁, IC₅₀: 1.7 nM (in human)	99.50%
Fiboflapon	LTB₄, IC₅₀: 76 nM						98.54%
LY223982	LTB₄, IC₅₀: 13.2 nM						99.67%
5-O-Demethylnobiletin		LTC₄, IC₅₀: 0.35 μM					99.93%
Veliflapon	LTB₄	LTC₄					99.48%
Fiboflapon sodium	LTB₄, IC₅₀: 76 nM						99.91%
Pranlukast		LTC₄, Ki: 5640 nM	LTD₄, Ki: 0.99 nM	LTE₄, Ki: 0.63 nM			98.18%
Nedocromil		LTC₄					98.02%
KP496			LTD₄				99.79%
Tipelukast			LTD₄, pA2: 6.41 (In guinea-pigs)	LTE₄, pA2: 6.45 (In guinea-pigs)			≥99.0%
Nedocromil sodium		LTC₄
(S)-Verapamil hydrochloride		LTC₄					99.39%
Amelubant	LTB₄, Ki: 221 nM (in vital human granulocytes) LTB₄, Ki: 230 nM (in cell membranes)						99.11%
AS-35		LTC₄, IC₅₀: 8 nM (In isolated guinea pig ileum)	LTD₄, IC₅₀: 4 nM (In isolated guinea pig ileum)	LTE₄, IC₅₀: 3 nM (In isolated guinea pig ileum)
Darbufelone mesylate	LTB₄						98.45%
Pranlukast hemihydrate		LTC₄, Ki: 5640 nM	LTD₄, Ki: 0.99 nM	LTE₄, Ki: 0.63 nM			99.28%
Quinotolast sodium		LTC₄					98.12%
Montelukast						CysLT₁
Montelukast dicyclohexylamine						CysLT₁
CAY10789						CysLT₁, IC₅₀: 2.80 ± 0.3 μM
DW-1350	LTB₄
CAY10583	LTB₄
HAMI 3379					CysLT₂
CP-96021 hydrochloride		LTC₄, Ki: 34 nM
CP-96486			LTD₄, Ki: 20 nM
Ablukast			LTD₄				99.36%
LM-1484		LTC₄	CysLT₁
RS-601			LTD₄
ONO4057	LTB₄, IC₅₀: 0.7 μM
LTD4 antagonist 1			LTD₄, Ki: 0.57 nM
LY210073	LTB₄, IC₅₀: 6.2 nM
CI-949		LTC₄, IC₅₀: 0.5 μM	LTD₄, IC₅₀: 0.5 μM
YM158 free base			LTD₄, pA2: 8.87
Bunaprolast	LTB₄
LTB4-IN-1	LTB₄, IC₅₀: 70 nM

Name
Email *

	Sorry, but the email address you supplied was invalid.