1. Signaling Pathways
  2. NF-κB
  3. NF-κB
  4. NF-κB Inhibitors

NF-κB Inhibitors

NF-κB

NF-κB1/p50

RelA/p65

RelB

c-Rel

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Please try each isoform separately.

NF-κB Inhibitors, Agonists, Activators, Modulators & Degraders
Product Name NF-κB NF-κB1/p50 RelA/p65 RelB c-Rel Purity
Phorbol 12-myristate 13-acetate
NF-κB
        99.80%
BAY 11-7082
NF-κB
        99.98%
JSH-23
NF-κB, IC50: 7.1 μM (in RAW 264.7 cells)
        99.92%
JP-11646
NF-κB
        98.74%
SAP15 acetate
NF-κB
 
p65
    98.04%
5-Aminosalicylic Acid    
p65
    99.97%
Baicalin
NF-κB
        98.92%
Shikonin
NF-κB
        99.80%
Sulfasalazine    
RelA
    99.57%
Pyrrolidinedithiocarbamate ammonium
NF-κB
        98.0%
TNF-α (31-45), human
NF-κB
        99.99%
Parthenolide
NF-κB
        99.91%
Fibrinogen (Bovine)  
p50
p65
 
c-Rel
Andrographolide  
p50
      99.74%
Withaferin A
NFκB
        99.92%
Betulinic acid
NF-κB
        99.88%
SC75741    
p65, IC50: 200 nM
    99.24%
Ginsenoside Rg1    
p65
    99.88%
20(S)-Ginsenoside Rg3    
p65
    99.82%
Nafamostat mesylate
I-kappaBalpha
        99.85%
Ginsenoside Rb1    
p65
    99.75%
Lidocaine
NF-κB
        99.96%
BAY 11-7085
NF-κB
        99.99%
(-)-DHMEQ    
RelA
RelB
  99.81%
NF-κΒ activator 1
NF-κB, EC50: 0.9 μM
        99.59%
α-Lipoic Acid
NF-κB
        99.94%
Diprovocim
NF-κB
        98.82%
Indole-3-carbinol
NF-κB
        99.16%
QNZ
NF-κB, IC50: 11 nM (in human Jurkat cells transfected with pNFκB-Luc)
        99.50%
CBL0137 hydrochloride
NF-κB, IC50: 0.47 μM
        99.72%
Caffeic acid phenethyl ester
NF-κB
        99.85%
Mangiferin  
p50
p65
    99.92%
Maslinic acid    
p65
    99.87%
Forsythoside B
NF-κB
        99.90%
MnTBAP chloride
NFκB
        98.0%
Saikosaponin D
NF-κB
        99.81%
Neferine    
p65
    99.92%
SN50
NF-κB
        99.62%
Astragalin    
p65
    99.94%
Isovitexin
NF-κB
        99.90%
Neochlorogenic acid    
p65
    99.80%
Lidocaine hydrochloride
NF-κB
        99.84%
18α-Glycyrrhetinic acid
NF-κB
        99.87%
Astilbin
NF-κB
        99.80%
Ginsenoside Re
NF-κB
        99.92%
Morusin    
p65
    99.54%
Vanillic acid    
p65
    99.75%
Tomatidine    
p65
    98.85%
Alendronic acid
NF-κB
        ≥98.0%
Okanin    
p65
    99.98%
Sinomenine hydrochloride
NF-κB
        99.89%
Stachydrine    
p65
    99.93%
EUK-134
NF-κB
        98.27%
Rhoifolin
NF-κB
        99.25%
Muscone
NF-κB
        98.0%
Anti-Mouse NK1.1 Antibody (PK136)
NF-κB
        98.57%
Nimbolide
NF-κB
        99.79%
Stachydrine hydrochloride    
p65
    99.90%
Ginsenoside Rd
NF-κB, IC50: 12.05 μM (in HepG2 cells)
        99.88%
DCZ0415
NF-κB
        99.81%
Guaiacol
NF-κB
        99.95%
(R)-Sulforaphane
NF-κB
        99.95%
Schisantherin A    
p65
    99.87%
Engeletin
NF-κB
        99.86%
Peimine
NFκB
        99.9%
Peiminine    
p65
    99.89%
NF-κΒ activator 2
NF-κB, EC50: 1.58 μM
        99.76%
Urocortin II, human
NF-κB
        99.95%
Oxaprozin
NF-κB
        99.94%
ASP-8731    
p65
    98.42%
Ethyl Caffeate
NF-κB
        99.34%
Sarsasapogenin
NF-κB
        99.93%
Ophiopogonin D
NF-κB
        99.80%
Licochalcone D    
p65
    99.80%
Plantainoside D
NF-κB
        99.15%
Lidocaine (Standard)
NF-κB
       
α-Lipoic Acid sodium
NF-κB
        99.95%
Anti-Mouse RANKL/CD254 Antibody (IK22/5)
NF-κB
        99.37%
Isobavachin
NF-κB
        99.88%
Chymostatin
NF-κB
        99.9%
Jolkinolide B
NFκB
        99.65%
Ginsenoside Rg5    
p65
    99.88%
Sciadopitysin
NF-κB
        99.0%
Ginsenoside Rb3
NF-κB, IC50: 8.2 μM (in 293T cell lines)
        99.87%
IT-901
NF-κB, IC50: 0.1 μM
     
c-Rel, IC50: 3 μM
99.32%
Myrcene,75% (stabilized with BHT)
NF-κB
       
2"-O-Galloylhyperin
NFκB
        99.57%
11-​Keto-​beta-​boswellic acid
NF-κB
        99.90%
Homoplantaginin    
p65
    99.90%
(±)-Naringenin
NF-κB
        99.83%
Ginsenoside Rg2
NF-κB
        98.71%
Hesperidin methylchalcone
NF-κB
        98.0%
CHPG
NF-κB
        99.51%
Lidocaine hydrochloride hydrate
NF-κB
        99.80%
Cafestol
NF-κB
        99.91%
Barlerin
NF-κB
        99.82%
Naringin Dihydrochalcone
NF-κB
        99.53%
CHPG sodium salt
NF-κB
        99.57%
Tenuigenin
NF-κB
        99.92%
Aconine
NF-κB
        99.81%
Deoxyelephantopin
NF-κB
        99.87%
Tectochrysin  
p50
p65
    99.88%
Tomatidine hydrochloride    
p65
    99.70%
Cynaropicrin
NF-κB
        99.79%
Ecliptasaponin A
NF-κB
        99.81%
Dendrophenol
NF-κB
        99.93%
L6H21
NF-κB
        99.19%
Sanggenon C
NF-κB
        98.46%
Sauchinone
I-kappaBalpha
 
p65
    99.62%
Yangonin    
RelA
    99.65%
Aurantiamide
NF-κB
        99.56%
2,5-Dihydroxyacetophenone
NF-κB
        99.95%
Inulicin
NF-κB
        99.94%
Cornuside
NF-κB
        99.99%
CDDO-dhTFEA
NF-κB
        99.64%
Ergolide    
p65
    99.48%
Triflusal
NF-κB
        99.56%
β-Funaltrexamine hydrochloride
NF-κB
        99.07%
Laquinimod
NF-κB
        99.46%
NF-κB/MAPK-IN-1
NF-κB
        98.71%
AT-533
NF-κB
        98.38%
Tianeptine
NF-κB
        99.84%
Polygalasaponin F
NF-κB
        99.85%
2'-Acetylacteoside
NF-κB
        99.73%
14-Deoxy-11,12-didehydroandrographolide
NF-κB
        99.93%
Reticuline
NF-κB
        98.89%
SM-7368
NF-κB
        99.77%
Ginsenoside Rk3
NF-κB, IC50: 14.24 μM (in HepG2 cells)
NF-κB, IC50: 15.32 μM (in SK-Hep1 cell)
        99.79%
N-(p-Coumaroyl) Serotonin
NF-κB
        99.03%
Isoliquiritin apioside
NF-κB
        99.87%
Cyclo(his-pro)
NF-κB
        98.95%
Chelidonic acid
NF-κB
        99.91%
JAK-IN-23
NF-κB, IC50: 150.7 nM
        98.88%
Armepavine
NF-κB
 
p65
    99.53%
Regaloside A    
p65
    99.64%
Rubiadin-1-methyl ether    
p65
    98.57%
Berubicin
NF-κB
       
(R)-(-)-Ibuprofen
NF-κB
        99.97%
Triacetylresveratrol
NF-κB
        99.11%
Obtusifolin
NF-κB
        99.91%
Methylthiouracil
NF-κB
        98.0%
Tianeptine sodium salt
NF-κB
        99.90%
4-O-Methyl honokiol
NF-κB
        98.76%
JP-163-16    
p65
    99.20%
Viridicatol
NF-κB
        99.93%
8-Deoxygartanin    
p65, IC50: 11.3 μM
    99.77%
Ginsenoside Rg6
NF-κB, IC50: 29.34 μM (in HepG2 cell)
NF-κB, IC50: 25.12 μM (in SK-Hep1 cell)
        99.87%
Cyclo(his-pro) TFA
NF-κB
        99.13%
Enniatin B1
NF-κB
        99.34%
Phenyl β-D-glucopyranoside
NF-κB
        99.85%
Ciwujianoside B
NF-κB
        99.68%
Ginsenoside F3
NF-κB
        99.84%
Urocortin II, human acetate
NF-κB
        99.61%
2′-Hydroxy-5′-methoxyacetophenone
NF-κB
        99.96%
CID-2858522
NF-κB, IC50: 70 nM
        99.78%
GlcNAc-MurNAc
NF-κB
       
Erdosteine
NF-κB
        99.54%
Anti-Mouse IL-9 Antibody (9C1)
NF-κB
       
Fosfenopril
NF-κB
        99.85%
NF-κB degrader 1  
p50
      99.92%
Quinocetone
NF-κB
        98.25%
Penehyclidine hydrochloride
NF-κB
        99.2%
Myricanol
NF-κB
        98.93%
Darutoside
NF-κB
        99.89%
PSP-0119
NF-κB
        98.65%
FIP22
NF-κB
        98.53%
Casuarinin
NF-κB
        98.24%
TNF-α (31-45), human TFA
NF-κB
        99.40%
MOR-106
NF-κB
       
Undecane
NF-κB
        99.66%
Anti-Mouse GITR Antibody (DTA-1)
NF-κB
        98.47%
Adelmidrol
NF-κB
        98.0%
DPLG3  
p50
p65
    99.18%
α-Lipoic Acid (Standard)
NF-κB
       
PROTAC STING degrader-4
NF-κB
        98.25%
RP-182
NF-κB
        98.68%
Hecogenin acetate
NF-κB
        98.57%
TML-6
NF-κB
        98.34%
Anemoside A3-methyl 6-aminohexanoate
NF-κB
        98.62%
Coelonin
NF-κB
        98.0%
Phellodendrine
NF-κB
        99.60%
Pellitorine
NF-κB
        99.84%
Flaconitine
NF-κB
        99.77%
Echinulin
NF-κB
        98.63%
Momordicine I
NF-κB
       
WAY-204688
NF-κB
        99.89%
Nafamostat
I-kappaBalpha
       
7,8-Dimethoxycoumarin
NF-κB
        99.75%
Salicortin
NF-κB
       
R-HP210
NF-κB
        98.21%
TAK-756
NF-κB
       
Sanggenon A
NF-κB
       
Anti-inflammatory agent 35
I-kappaBalpha
NF-κB
 
p65
    99.77%
Anemarsaponin B    
p65
    99.43%
Ginsenoside Rb1 (Standard)    
p65
   
Vitisin A
NF-κB
       
β-Patchoulene
NF-κB
       
SMU-14a    
p65
   
BRD4-BD1/2-IN-3    
p65
    99.52%
Gaultherin
NF-κB
        99.44%
Nafamostat hydrochloride
I-kappaBalpha
       
6-Methoxymellein
NF-κB
       
Laquinimod sodium
NF-κB
       
Anti-inflammatory agent 99
NF-κB
       
Penehyclidine
NF-κB
       
CIAC101
NF-κB
       
JWX-A0108
NF-κB
       
Mumefural
NF-κB
       
IMD-biphenylC
NF-κB
       
NF-κB-IN-3
NF-κB, IC50: 0.70 μM
       
Verproside
NF-κB
       
Ginsenoside Rb3 (Standard)
NF-κB
       
G721-0282
NF-κB
        99.96%
IAV-IN-5
NF-κB
       
IKKβ-IN-7    
p65
   
PROTAC HDAC6 degrader 7
NF-κB
       
MMH-165-26    
p65
   
Esculeogenin A
NF-κB
       
Acutissimalignan B
I-kappaBalpha
 
p65
   
SAP15
NF-κB
 
RelA
   
EC-70124
NF-κB
       
SHP2-IN-45
NF-κB
       
Ginsenoside Rd (Standard)
NF-κB
       
6-O-p-Hydroxybenzoylglutinoside
NF-κB, IC50: 52.78 μM
       
GNE-5472
NF-κB
       
CKD-712
NF-κB
       
Ephemeranthol A
NF-κB
       
Eudebeiolide B
NF-κB
       
DNH28
NF-κB
       
Ginsenoside Re (Standard)
NF-κB
       
Oxaprozin potassium
NF-κB
       
IMD-catechol
NF-κB
       
Sootepin D
NF-κB
       
BAY-356
NF-κB
       
G721-0377
NF-κB
       
NF-κB-IN-14
NF-κB
       
TP-110
NF-κB
       
STAT3/NF-κB-IN-1
NF-κB, IC50: 4.22 μM
       
XRF-1021
NF-κB
       
Lucidone
NF-κB
p50
p65
   
MEDI-5083
NF-κB
       
Bartogenic acid
NF-κB
       
Orazipone
NF-κB
       
N,N-Diethylacetamide
NF-κB
        99.68%
Cannabitwinol
NF-κB
       
IMD-biphenylB
NF-κB
       
Aurothiomalate disodium
NF-κB
       
Panaxytriol
NF-κB
       
TKL002
NF-κB
       
Anti-inflammatory agent 20
NF-κB
       
Coronalolic acid
NF-κB
       
Ginsenoside Rg2 (Standard)
NF-κB
       
MR2938
NF-κB
       
Xanthine oxidase-IN-6
NF-κB
       
Urocortin II, human TFA
NF-κB
       
LM9
NF-κB
       
β-Funaltrexamine
NF-κB
       
20(S)-Ginsenoside Rg3 (Standard)    
p65
   
NLRP3-IN-32    
p65
   
Mesalamine impurity P
NF-κB
       
Dth  
p50
p65
   
Triphala
NF-κB
       
HDAC6-IN-71
NF-κB
       
PPARγ agonist-21
NF-κB
       
NIK-IN-3
NF-κB, IC50: 5.2 nM
       
Triptolidenol    
p65
   
GUT-70
NF-κB
       
Ginsenoside Rg1 (Standard)    
p65
   
CAY10512
NF-κB
       
Triflusal-d3
NF-κB
       
Jolkinolide B (Standard)
NF-κB
       
Anti-inflammatory agent 107
NF-κB
       
Cudraflavone B
NF-κB
       
CLP-d2
I-kappaBalpha
 
p65
   
sEH-IN-21
NF-κB
       
NF-κB-IN-20
NF-κB
       
RIPK1-IN-32
NF-κB
       
2'-Acetylacteoside (Standard)
NF-κB
       
Xanthine oxidase-IN-21
NF-κB
       
4-Methoxycinnamic acid ethyl ester
NF-κB, IC50: 88.7 μM
       
Glycoursodeoxycholic acid 3-sulfate    
p65
   
Triflusal (Standard)
NF-κB
       
N-(p-Coumaroyl) Serotonin (Standard)
NF-κB
       
(S)-(-)-Anatabine
NF-κB
       
DHMEQ racemate
NF-κB
       
Acetoxycycloheximide
NF-κB
       
NF-κB-IN-13
NF-κB
       
Anti-Mouse Delta-like protein 4/DLL4 Antibody (HMD4-2)
NF-κB
       
Berkeleyacetal C
NF-κB
       
2"-O-Galloylhyperin (Standard)
NF-κB
       
Icariside F2
NF-κB, IC50: 16.25 μM