2. GPCR/G Protein
  3. P2Y Receptor
  4. Becondogrel

Becondogrel  (Synonyms: 2-Oxoclopidogrel)

Cat. No.: HY-172417 Purity: 99.39% ee.: 99.12%
COA
SDS
Handling Instructions Technical Support

Becondogrel (2-Oxoclopidogrel) is the metabolite of Clopidogrel (HY-15283). Becondogrel irreversibly inhibits P2Y12 receptor, thereby inhibiting platelet aggregation and thrombosis.

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Becondogrel

Becondogrel 화학구조

CAS No. : 1416696-44-0

사이즈 가격 재고 수량
5 mg 해외재고보유
10 mg   견적 받기  
50 mg   견적 받기  

* 장바구니에 담기 전 물품의 수량을 선택해 주십시오.

This product is a controlled substance and not for sale in your territory.

고객리뷰

Based on 1 Customer Validation

Becondogrel Related Antibodies

Top Publications Citing Use of Products

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P2Y1 Receptor P2Y2 Receptor P2Y6 Receptor P2Y11 Receptor P2Y12 Receptor P2Y13 Receptor P2Y14 Receptor

  • Biological Activity

  • 순도&문서

  • References

  • 고객리뷰

제품 설명

Becondogrel (2-Oxoclopidogrel) is the metabolite of Clopidogrel (HY-15283). Becondogrel irreversibly inhibits P2Y12 receptor, thereby inhibiting platelet aggregation and thrombosis[1].

분자량

337.82

화학식

C16H16ClNO3S
CAS No.
Appearance

Solid

Color

White to off-white

SMILES

COC([C@H](C1=C(C=CC=C1)Cl)N2CC([C@](S3)([H])CC2)=CC3=O)=O
선적

Room temperature in continental US; may vary elsewhere.
보관
Powder -20°C 3 years
4°C 2 years
In solvent -80°C 6 months
-20°C 1 month
용액&용해도
In Vitro: 

DMSO : 60 mg/mL (177.61 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.9602 mL 14.8008 mL 29.6016 mL
5 mM 0.5920 mL 2.9602 mL 5.9203 mL
View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

  • 몰농도 계산기

  • 농도 희석 계산기

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass
=
Concentration
×
Volume
×
Molecular Weight *

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start)

C1

×
Volume (start)

V1

=
Concentration (final)

C2

×
Volume (final)

V2

In Vivo Dissolution Calculator
Please enter the basic information of animal experiments:

Dosage

mg/kg

Animal weight
(per animal)

g

Dosing volume
(per animal)

μL

Number of animals

Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.
Calculation results:
Working solution concentration: mg/mL
순도&문서
References

Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

Optional Solvent Concentration Solvent Mass 1 mg 5 mg 10 mg 25 mg
DMSO 1 mM 2.9602 mL 14.8008 mL 29.6016 mL 74.0039 mL
5 mM 0.5920 mL 2.9602 mL 5.9203 mL 14.8008 mL
10 mM 0.2960 mL 1.4801 mL 2.9602 mL 7.4004 mL
15 mM 0.1973 mL 0.9867 mL 1.9734 mL 4.9336 mL
20 mM 0.1480 mL 0.7400 mL 1.4801 mL 3.7002 mL
25 mM 0.1184 mL 0.5920 mL 1.1841 mL 2.9602 mL
30 mM 0.0987 mL 0.4934 mL 0.9867 mL 2.4668 mL
40 mM 0.0740 mL 0.3700 mL 0.7400 mL 1.8501 mL
50 mM 0.0592 mL 0.2960 mL 0.5920 mL 1.4801 mL
60 mM 0.0493 mL 0.2467 mL 0.4934 mL 1.2334 mL
80 mM 0.0370 mL 0.1850 mL 0.3700 mL 0.9250 mL
100 mM 0.0296 mL 0.1480 mL 0.2960 mL 0.7400 mL
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Becondogrel Related Classifications

Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Becondogrel1416696-44-02-OxoclopidogrelP2Y ReceptorInhibitorinhibitorinhibit

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상품명:
Becondogrel
Cat. No.:
HY-172417
수량:
MCE Japan Authorized Agent:

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SAFETY DATA SHEET (SDS)

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