1052515-91-9

VU0134992 hydrochloride Chemical Structure
1052515-91-9

Chemical Structure

VU0134992 hydrochloride

  • CAS No.: 1052515-91-9
  • Formula:C20H32BrClN2O2
  • Molecular Weight:447.84

IUPAC Name: 2-(2-bromo-4-isopropylphenoxy)-N-(2,2,6,6-tetramethylpiperidin-4-yl)acetamide hydrochloride

InChIKey: QXKQUPCNSXWIDX-UHFFFAOYSA-N

SMILES: O=C(NC1CC(C)(C)NC(C)(C)C1)COC2=CC=C(C(C)C)C=C2Br.[H]Cl

Biological Activity: VU0134992 hydrochloride is the first subtype-preferring, orally active and selective Kir4.1 potassium channel pore blocker, with an IC50 of 0.97 µM. VU0134992 hydrochloride is 9-fold selective for homomeric Kir4.1 over Kir4.1/5.1 concatemeric channels (IC50=9 µM) at -120 mV[1].

Cat. No. Product Name Purity Description Pricing
HY-122560A 		VU0134992 hydrochloride 98.49% VU0134992 hydrochloride is the first subtype-preferring, orally active and selective Kir4.1 potassium channel pore blocker, with an IC50 of 0.97 µM. VU0134992 hydrochloride is 9-fold selective for homomeric Kir4.1 over Kir4.1/5.1 concatemeric channels (IC50=9 µM) at -120 mV.
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