105878-43-1
105878-43-1
Chemical Structure
Bisoprolol fumarate
- CAS No.: 105878-43-1
- Formula:C22H35NO8
- Molecular Weight:441.52
IUPAC Name: 1-(4-((2-isopropoxyethoxy)methyl)phenoxy)-3-(isopropylamino)propan-2-ol fumarate
InChIKey: RZPZLFIUFMNCLY-WLHGVMLRSA-N
SMILES: OC(COC1=CC=C(C=C1)COCCOC(C)C)CNC(C)C.OC(/C=C/C(O)=O)=O
Biological Activity: Bisoprolol fumarate is a potent, selective and orally active β1-adrenergic receptor blocker with little activity on β2-receptor. Bisoprolol fumarate has the potential for hypertension, coronary artery disease and stable ventricular dysfunction research[1][2].
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Bisoprolol fumarate | Bisoprolol fumarate is a potent, selective and orally active β1-adrenergic receptor blocker with little activity on β2-receptor. Bisoprolol fumarate has the potential for hypertension, coronary artery disease and stable ventricular dysfunction research. | |||||||||||||||||||||
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Bisoprolol-d5 hemifumarate | Bisoprolol-d5 (hemifumarate) is deuterium labeled Bisoprolol (fumarate). | |||||||||||||||||||||
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References
- [1]. Jillian G Baker, et al. The selectivity of beta-adrenoceptor antagonists at the human beta1, beta2 and beta3 adrenoceptors. Br J Pharmacol. 2005 Feb;144(3):317-22. [Content Brief]
- [2]. Jing Wang, et al. Bisoprolol, a β 1 antagonist, protects myocardial cells from ischemia-reperfusion injury via PI3K/AKT/GSK3β pathway. Fundam Clin Pharmacol. 2020 Dec;34(6):708-720. [Content Brief]
