1124167-61-8
Chemical Structure
Mu opioid receptor antagonist 5
- CAS No.: 1124167-61-8
- Formula:C26H29N3O4
- Molecular Weight:447.53
IUPAC Name: N-((4R,4aS,7R,7aR,12bS)-3-(cyclopropylmethyl)-4a,9-dihydroxy-2,3,4,4a,5,6,7,7a-octahydro-1H-4,12-methanobenzofuro[3,2-e]isoquinolin-7-yl)isonicotinamide
InChIKey: XQWZTPWKACKUMJ-HJUABUFYSA-N
SMILES: O[C@]12[C@H]3CC4=C5[C@@]1(CCN3CC6CC6)[C@H]([C@@H](CC2)NC(C7=CC=NC=C7)=O)OC5=C(O)C=C4
Biological Activity: Mu opioid receptor antagonist 5 (compound NAP) is a selective and blood-brain barrier (BBB) penetrant μ opioid receptor (MOR) antagonist with an EC50 value of 1.14 nM and a Ki value of 0.37 nM. Mu opioid receptor antagonist 5 can be used for researching opioid use disorders (OUD)[1].
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Mu opioid receptor antagonist 5 | Mu opioid receptor antagonist 5 (compound NAP) is a selective and blood-brain barrier (BBB) penetrant μ opioid receptor (MOR) antagonist with an EC50 value of 1.14 nM and a Ki value of 0.37 nM. Mu opioid receptor antagonist 5 can be used for researching opioid use disorders (OUD). | |||||||||||||||||||||
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Keywords
