1189805-13-7
Chemical Structure
Molindone-d8
Synonym(s): (±)-Molindone-d8;SPN-810M-d8
- CAS No.: 1189805-13-7
- Formula:C16H16D8N2O2
- Molecular Weight:284.42
IUPAC Name: 3-ethyl-2-methyl-5-((morpholino-d8)methyl)-1,5,6,7-tetrahydro-4H-indol-4-one
InChIKey: KLPWJLBORRMFGK-COMRDEPKSA-N
SMILES: C(C)C=1C2=C(NC1C)CCC(CN3C(C(OC(C3([2H])[2H])([2H])[2H])([2H])[2H])([2H])[2H])C2=O
Biological Activity: Molindone-d8 is the deuterium labeled Molindone. Molindone hydrochloride (EN-1733A) is a therapeutic antipsychotic, used in the treatment of schizophrenia, works by blocking the effects of dopamine in the brain, leading to diminished psychoses[1][2].
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Molindone-d8 | 99.2% | Molindone-d8 is the deuterium labeled Molindone. Molindone hydrochloride (EN-1733A) is a therapeutic antipsychotic, used in the treatment of schizophrenia, works by blocking the effects of dopamine in the brain, leading to diminished psychoses. | ||||||||||||||||||||
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Molindone | Molindone ((±)-Molindone), an indole derivative, is a potent dopamine D2 and D5 receptor antagonist. Molindone ((±)-Molindone) can be used for the research of schizophrenia and severe mental illness. | |||||||||||||||||||||
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- [1]. Yu C, et al. In vitro pharmacological characterization of SPN-810M (molindone). J Exp Pharmacol. 2018;10:65-73. Published 2018 Nov 21. [Content Brief]
- [2]. Russak EM, et al. Impact of Deuterium Substitution on the Pharmacokinetics of Pharmaceuticals. Ann Pharmacother. 2019;53(2):211-216. [Content Brief]
Keywords
