1346747-40-7
1346747-40-7
Chemical Structure
(±)-Penbutolol-d9
Synonym(s): (Rac)-Penbutolol-d9;(±)-Isopenbutolol-d9
- CAS No.: 1346747-40-7
- Formula:C18H20D9NO2
- Molecular Weight:300.48
IUPAC Name: 1-(2-cyclopentylphenoxy)-3-((2-(methyl-d3)propan-2-yl-1,1,1,3,3,3-d6)amino)propan-2-ol
InChIKey: KQXKVJAGOJTNJS-GQALSZNTSA-N
SMILES: OC(CNC(C([2H])([2H])[2H])(C([2H])([2H])[2H])C([2H])([2H])[2H])COC1=CC=CC=C1C2CCCC2
Biological Activity: (±)-Penbutolol-d9 is the deuterium labeled (±)-Penbutolol[1].
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(±)-Penbutolol-d9 | (±)-Penbutolol-d9 is the deuterium labeled (±)-Penbutolol. | |||||||||||||||||||||
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(±)-Penbutolol-d9 hydrochloride | (±)-Penbutolol-d9 (hydrochloride) is a deuterium labeled (±)-Penbutolol hydrochloride. (+)-Penbutolol hydrochloride is a β-adrenoceptor antagonist, with an IC50 of 0.74 μM. | |||||||||||||||||||||
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(±)-Penbutolol | 98.07% | (±)-Penbutolol ((Rac)-Penbutolol) is the racemic mixture of Penbutolol. (±)-Penbutolol is an orally active β-adrenergic receptor antagonist. (±)-Penbutolol antagonizes exercise-induced tachycardia, reduces the increase in peak expiratory flow rate (PEFR) caused by exercise, and decreases resting plasma renin activity (PRA). (±)-Penbutolol reaches peak plasma concentration 1 hour after oral administration, with a half-life of 4.5 hours, and is converted into an active metabolite in the body. (±)-Penbutolol can be used in cardiovascular-related disease research. | ||||||||||||||||||||
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References
