1400811-63-3
1400811-63-3
Chemical Structure
PF-03382792
- CAS No.: 1400811-63-3
- Formula:C23H32FN3O4
- Molecular Weight:433.52
IUPAC Name: 6-fluoro-N-((1-((4-hydroxytetrahydro-2H-pyran-4-yl)methyl)piperidin-4-yl)methyl)-3,3-dimethyl-2-oxoindoline-1-carboxamide
InChIKey: AGMOFKKOVMRGAK-UHFFFAOYSA-N
SMILES: O=C(N1C(C(C)(C)C2=C1C=C(F)C=C2)=O)NCC3CCN(CC4(O)CCOCC4)CC3
Biological Activity: PF-03382792 is a potent 5-HT4 partial agonist with a Ki of 2.7 nM and an EC50 of 0.9 nM for 5-HT4d. PF-03382792 can penetrate the brain. PF-03382792 produces moderate increases in cortical Ach in the rat prefrontal cortex[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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PF-03382792 | 99.58% | PF-03382792 is a potent 5-HT4 partial agonist with a Ki of 2.7 nM and an EC50 of 0.9 nM for 5-HT4d. PF-03382792 can penetrate the brain. PF-03382792 produces moderate increases in cortical Ach in the rat prefrontal cortex. | ||||||||||||||||||||
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References
Keywords
