141636-65-9
141636-65-9
Chemical Structure
GR 94800
- CAS No.: 141636-65-9
- Formula:C49H61N9O8
- Molecular Weight:904.06
SMILES: [Bz-AA-{D-Trp}-F-{D-Pro}-P-{Nle}-NH2]
Biological Activity: GR 94800 is a potent and selective NK2 receptor peptide antagonist, with pKB values of 9.6, 6.4 and 6.0 for NK2, NK1 and NK3 receptors, respectively[1][2].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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GR 94800 | 99.42% | GR 94800 is a potent and selective NK2 receptor peptide antagonist, with pKB values of 9.6, 6.4 and 6.0 for NK2, NK1 and NK3 receptors, respectively. | ||||||||||||||||||||
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References
- [1]. A B McElroy, et al. Highly potent and selective heptapeptide antagonists of the neurokinin NK-2 receptor. J Med Chem. 1992 Jul 10;35(14):2582-91. [Content Brief]
- [2]. M A Matuszek, et al. An investigation of tachykinin NK2 receptor subtypes in the rat. Eur J Pharmacol. 1998 Jul 3;352(1):103-9. [Content Brief]
Keywords
