1. GPCR/G Protein
    Neuronal Signaling
  2. Neurokinin Receptor
  3. GR 94800

GR 94800 

Cat. No.: HY-P1277
Handling Instructions

GR 94800 is a potent and selective NK2 receptor peptide antagonist, with pKB values of 9.6, 6.4 and 6.0 for NK2, NK1 and NK3 receptors, respectively.

For research use only. We do not sell to patients.

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GR 94800 Chemical Structure

GR 94800 Chemical Structure

CAS No. : 141636-65-9

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Description

GR 94800 is a potent and selective NK2 receptor peptide antagonist, with pKB values of 9.6, 6.4 and 6.0 for NK2, NK1 and NK3 receptors, respectively[1][2].

In Vitro

Responses to EFS (15 Hz) were significantly reduced by the NK2 receptor antagonist GR 94800 (1 μM) either alone or in combination with the NK1 antagonist (1 μM)[3].

Molecular Weight

904.06

Formula

C₄₉H₆₁N₉O₈

CAS No.

141636-65-9

Sequence Shortening

Bz-AA-{D-Trp}-F-{D-Pro}-P-{Nle}-NH2

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Keywords:

GR 94800GR94800GR-94800Neurokinin ReceptorNK receptorInhibitorinhibitorinhibit

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GR 94800
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