1. GPCR/G Protein
    Neuronal Signaling
  2. Neurokinin Receptor
  3. GR 94800 TFA

GR 94800 TFA 

Cat. No.: HY-P1277A
Handling Instructions

GR 94800 TFA is a potent and selective NK2 receptor peptide antagonist, with pKB values of 9.6, 6.4 and 6.0 for NK2, NK1 and NK3 receptors, respectively.

For research use only. We do not sell to patients.

Custom Peptide Synthesis

GR 94800 TFA Chemical Structure

GR 94800 TFA Chemical Structure

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Description

GR 94800 TFA is a potent and selective NK2 receptor peptide antagonist, with pKB values of 9.6, 6.4 and 6.0 for NK2, NK1 and NK3 receptors, respectively[1][2].

In Vitro

Responses to EFS (15 Hz) were significantly reduced by the NK2 receptor antagonist GR 94800 (1 μM) either alone or in combination with the NK1 antagonist (1 μM)[3].

Molecular Weight

1018.08

Formula

C₅₁H₆₂F₃N₉O₁₀

Sequence Shortening

Bz-AA-{D-Trp}-F-{D-Pro}-P-{Nle}-NH2

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
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Keywords:

GR 94800GR94800GR-94800Neurokinin ReceptorNK receptorInhibitorinhibitorinhibit

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GR 94800 TFA
Cat. No.:
HY-P1277A
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