1593478-56-8
1593478-56-8
Chemical Structure
(R)-CE3F4
- CAS No.: 1593478-56-8
- Formula:C11H10Br2FNO
- Molecular Weight:351.01
IUPAC Name: (R)-5,7-dibromo-6-fluoro-2-methyl-3,4-dihydroquinoline-1(2H)-carbaldehyde
InChIKey: ZZLQPWXVZCPUGC-ZCFIWIBFSA-N
SMILES: O=CN1[C@H](C)CCC2=C1C=C(Br)C(F)=C2Br
Biological Activity: (R)-CE3F4 is a potent and selective inhibitor of exchange protein directly activated by cAMP isoform 1 (Epac1), with an IC50 of 4.2 μM, with 10-fold selectivity for Epac1 over Epac2 (IC50, 44 μM). (R)-CE3F4 is more potent than racemic CE3F4 and (S)-CE3F4[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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(R)-CE3F4 | 99.3% | (R)-CE3F4 is a potent and selective inhibitor of exchange protein directly activated by cAMP isoform 1 (Epac1), with an IC50 of 4.2 μM, with 10-fold selectivity for Epac1 over Epac2 (IC50, 44 μM). (R)-CE3F4 is more potent than racemic CE3F4 and (S)-CE3F4. | ||||||||||||||||||||
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References
Keywords
