1629277-36-6
1629277-36-6
Chemical Structure
PNZ5
- CAS No.: 1629277-36-6
- Formula:C20H18N2O2
- Molecular Weight:318.37
IUPAC Name: (S)-5-(3,5-dimethylisoxazol-4-yl)-2-methyl-3-phenylisoindolin-1-one
InChIKey: CHAKVDDAHQGTLR-IBGZPJMESA-N
SMILES: CN1C(C2=CC=C(C3=C(C)ON=C3C)C=C2[C@@]1(C4=CC=CC=C4)[H])=O
Biological Activity: PNZ5 is a potent and isoxazole-based pan-BET inhibitor with high selectivity and potency similar to the well-established (+)-JQ1, with a KD of 5.43 nM for BRD4(1)[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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PNZ5 | 99.61% | PNZ5 is a potent and isoxazole-based pan-BET inhibitor with high selectivity and potency similar to the well-established (+)-JQ1, with a KD of 5.43 nM for BRD4(1). | ||||||||||||||||||||
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References
Keywords
