1648726-56-0
1648726-56-0
Chemical Structure
PF-04781340
- CAS No.: 1648726-56-0
- Formula:C17H21N3
- Molecular Weight:267.37
IUPAC Name: 3-benzyl-N-methyl-6,7,8,9-tetrahydro-5H-pyrido[3,4-d]azepin-1-amine
InChIKey: HFAURKSQTSLTBO-UHFFFAOYSA-N
SMILES: CNC1=NC(CC2=CC=CC=C2)=CC3=C1CCNCC3
Biological Activity: PF-04781340 is a potent and selective 5-HT2C receptor agonist, with an EC50 of 9 nM and a Ki of 3 nM, respectively. PF-04781340 exhibits weak partial agonist activity at the 5-HT2B receptor, with an EC50 of 1484 nM. PF-04781340 can be used in the research of obesity and psychiatric disorders[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
|
|
PF-04781340 | PF-04781340 is a potent and selective 5-HT2C receptor agonist, with an EC50 of 9 nM and a Ki of 3 nM, respectively. PF-04781340 exhibits weak partial agonist activity at the 5-HT2B receptor, with an EC50 of 1484 nM. PF-04781340 can be used in the research of obesity and psychiatric disorders. | |||||||||||||||||||||
|
loading...
/
|
|||||||||||||||||||||||
References
Keywords
