1875078-61-7
1875078-61-7
Chemical Structure
BCAT-IN-1
- CAS No.: 1875078-61-7
- Formula:C25H24BrN5O2S
- Molecular Weight:538.46
IUPAC Name: 1-((1R,3S)-3-(5-bromothiophene-2-carboxamido)cyclohexyl)-N-methyl-2-(pyridin-2-yl)-1H-benzo[d]imidazole-5-carboxamide
InChIKey: PGSKODUPOMCUEJ-DLBZAZTESA-N
SMILES: O=C(C1=CC=C2N([C@H]3C[C@@H](NC(C4=CC=C(Br)S4)=O)CCC3)C(C5=NC=CC=C5)=NC2=C1)NC
Biological Activity: BCAT-IN-1 is a potent, selective and orally active inhibitor of BCATm, with a pIC50 of 7.3. BCAT-IN-1 shows 100-fold selectivity for BCATm over BCATc (pIC50=5.4). BCAT-IN-1 can be used for the research of metabolic diseases[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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BCAT-IN-1 | 98.06% | BCAT-IN-1 is a potent, selective and orally active inhibitor of BCATm, with a pIC50 of 7.3. BCAT-IN-1 shows 100-fold selectivity for BCATm over BCATc (pIC50=5.4). BCAT-IN-1 can be used for the research of metabolic diseases. | ||||||||||||||||||||
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References
Keywords
