1953134-15-0
1953134-15-0
Chemical Structure
(1S,3R)-GNE-502
- CAS No.: 1953134-15-0
- Formula:C25H30FN3O3S
- Molecular Weight:471.59
IUPAC Name: (1S,3R)-1-(4-(2-(3-(fluoromethyl)azetidin-1-yl)ethoxy)phenyl)-3-methyl-2-(methylsulfonyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole
InChIKey: ALLRPIPLWLLBGX-NSYGIPOTSA-N
SMILES: C[C@@H]1CC(C2=CC=CC=C2N3)=C3[C@H](C4=CC=C(C=C4)OCCN5CC(C5)CF)N1S(=O)(C)=O
Biological Activity: (1S,3R)-GNE-502 (compound 179) is a potent ERα degrader with an EC50 value of 13 nM against ERα in MCF7 HCS. (1S,3R)-GNE-502 can be used to research cancer related with estrogen receptor[1].
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(1S,3R)-GNE-502 | (1S,3R)-GNE-502 (compound 179) is a potent ERα degrader with an EC50 value of 13 nM against ERα in MCF7 HCS. (1S,3R)-GNE-502 can be used to research cancer related with estrogen receptor. | |||||||||||||||||||||
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References
Keywords
