214348-67-1
Chemical Structure
L-054522
- CAS No.: 214348-67-1
- Formula:C35H47N7O5
- Molecular Weight:645.79
IUPAC Name: tert-butyl ((2R,3S)-3-(1H-indol-3-yl)-2-(4-(2-oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)piperidine-1-carboxamido)butanoyl)-L-lysinate
InChIKey: WFCIXKAZBUIFTR-PKIMSIDOSA-N
SMILES: O=C([C@H](CCCCN)NC([C@@H]([C@@H](C)C1=CNC2=C1C=CC=C2)NC(N3CCC(CC3)N4C5=CC=CC=C5NC4=O)=O)=O)OC(C)(C)C
Biological Activity: L-054522 is an agonist for somatostatin receptor subtype 2 with Kd of 0.01 nM. L-054522 inhibits growth hormone release from rat primary pituitary cell (IC50=0.05 nM) and glucagon and insulin release from isolated mouse pancreatic islet cell (IC50=0.05 nM and 12 nM)[1].
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L-054522 | L-054522 is an agonist for somatostatin receptor subtype 2 with Kd of 0.01 nM. L-054522 inhibits growth hormone release from rat primary pituitary cell (IC50=0.05 nM) and glucagon and insulin release from isolated mouse pancreatic islet cell (IC50=0.05 nM and 12 nM). | |||||||||||||||||||||
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Keywords
