2171386-10-8
2171386-10-8
Chemical Structure
RK-287107
- CAS No.: 2171386-10-8
- Formula:C22H26F2N4O2
- Molecular Weight:416.46
IUPAC Name: 2-(4,6-difluoro-1-(2-hydroxyethyl)spiro[indoline-3,4'-piperidin]-1'-yl)-5,6,7,8-tetrahydroquinazolin-4(3H)-one
InChIKey: FZQYCOUBRJEYBC-UHFFFAOYSA-N
SMILES: O=C1NC(N2CCC3(CC2)CN(CCO)C4=C3C(F)=CC(F)=C4)=NC5=C1CCCC5
Biological Activity: RK-287107 is a potent and specific tankyrase inhibitor with IC50s of 14.3 and 10.6 nM for tankyrase-1 and tankyrase-2, respectively. RK-287107 blocks colorectal cancer cell growth[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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RK-287107 | 99.80% | RK-287107 is a potent and specific tankyrase inhibitor with IC50s of 14.3 and 10.6 nM for tankyrase-1 and tankyrase-2, respectively. RK-287107 blocks colorectal cancer cell growth. | ||||||||||||||||||||
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References
Keywords
