2242428-57-3
Chemical Structure
Elunonavir
- CAS No.: 2242428-57-3
- Formula:C52H59F10N11O8
- Molecular Weight:1156.08
InChIKey: ZTSLYWLHCOINNI-FTEFBJIISA-N
SMILES: O=C(N[C@@H](CC1=CC=C(C#CC2=CN=C(N=C2)N3CC4CCC(C3)N4C5COC5)C=C1)[C@H](CN(CC(C(F)=C6)=C(F)C=C6C7=NN(C(F)F)C=C7)NC([C@@H](NC(OC)=O)C(C)(C(F)(F)F)C)=O)O)[C@@H](NC(OC)=O)C(C)(C(F)(F)F)C
Biological Activity: Elunonavir (GS-1156) is a HIV protease inhibitor with a high barrier to resistance and excellent metabolic stability. Elunonavir is able to overcome rapid CYP-mediated metabolism, resulting in a significantly prolonged half-life and the potential to reduce dosing frequency without the need for pharmacokinetic enhancers[1].
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Elunonavir | Elunonavir (GS-1156) is a HIV protease inhibitor with a high barrier to resistance and excellent metabolic stability. Elunonavir is able to overcome rapid CYP-mediated metabolism, resulting in a significantly prolonged half-life and the potential to reduce dosing frequency without the need for pharmacokinetic enhancers. | |||||||||||||||||||||
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Keywords
