244101-02-8
244101-02-8
Chemical Structure
L-798106
Synonym(s): CM9; GW671021
- CAS No.: 244101-02-8
- Formula:C27H22BrNO4S
- Molecular Weight:536.44
IUPAC Name: (E)-N-((5-bromo-2-methoxyphenyl)sulfonyl)-3-(2-(naphthalen-2-ylmethyl)phenyl)acrylamide
InChIKey: ODTKFNUPVBULRJ-NTCAYCPXSA-N
SMILES: O=C(NS(=O)(C1=CC(Br)=CC=C1OC)=O)/C=C/C2=CC=CC=C2CC3=CC=C4C=CC=CC4=C3
Biological Activity: L-798106 is potent and highly selective prostanoid EP3 receptor antagonist (Ki=0.3 nM), it also has micromolar activities at the EP4, EP1 and EP2 receptors with Ki values of 916 nM, >5000 nM and >5000 nM, respectively[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
|
|
L-798106 | 99.91% | L-798106 is potent and highly selective prostanoid EP3 receptor antagonist (Ki=0.3 nM), it also has micromolar activities at the EP4, EP1 and EP2 receptors with Ki values of 916 nM, >5000 nM and >5000 nM, respectively. | ||||||||||||||||||||
|
loading...
/
|
|||||||||||||||||||||||
References
Keywords
