2507890-46-0
Chemical Structure
LuAF60097
- CAS No.: 2507890-46-0
- Formula:C32H32FN3O3
- Molecular Weight:525.62
IUPAC Name: (S)-1-(4-fluorophenyl)-1-(3-(4-(2-oxo-1,2-dihydroquinolin-7-yl)piperidin-1-yl)propyl)-1,3-dihydroisobenzofuran-5-carboxamide
InChIKey: KNQRTZFUQPXVLO-YTTGMZPUSA-N
SMILES: C(CCN1CCC(CC1)C=2C=C3C(=CC2)C=CC(=O)N3)[C@@]4(C=5C(CO4)=CC(C(N)=O)=CC5)C6=CC=C(F)C=C6
Biological Activity: LuAF60097 is a serotonin transporter (SERT) ligand. LuAF60097 binds to the extracellular vestibule (S2 site) of SERT with high affinity and to the central binding site (S1) with lower affinity, triggering conformational changes that exert combined competitive and non-competitive inhibitory effects on serotonin reuptake. LuAF60097 is applicable to research related to depression and anxiety disorders[1].
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LuAF60097 | LuAF60097 is a serotonin transporter (SERT) ligand. LuAF60097 binds to the extracellular vestibule (S2 site) of SERT with high affinity and to the central binding site (S1) with lower affinity, triggering conformational changes that exert combined competitive and non-competitive inhibitory effects on serotonin reuptake. LuAF60097 is applicable to research related to depression and anxiety disorders. | |||||||||||||||||||||
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