2655557-54-1
2655557-54-1
Chemical Structure
ITK/TRKA-IN-1
- CAS No.: 2655557-54-1
- Formula:C25H30F2N6O2
- Molecular Weight:484.54
IUPAC Name: (S)-N-(2-((4aS,5aR)-5,5-difluoro-5a-methyl-1,4,4a,5,5a,6-hexahydrocyclopropa[f]indazol-3-yl)-6-methyl-1H-benzo[d]imidazol-5-yl)-N-methyl-2-morpholinopropanamide
InChIKey: PWTZWYZDFORBCV-OSZRXVRWSA-N
SMILES: C[C@@]12CC3=C(C(C4=NC5=C(N4)C=C(C(N(C([C@@H](N6CCOCC6)C)=O)C)=C5)C)=NN3)C[C@@H]1C2(F)F
Biological Activity: ITK/TRKA-IN-1 is a dual inhibitor of IL-2-inducible T-cell kinase (ITK) and tropomyosin receptor kinase A (TRKA) with an IC50 value of 1.0 nM and 96 % inhibition, respectively.
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ITK/TRKA-IN-1 | ITK/TRKA-IN-1 is a dual inhibitor of IL-2-inducible T-cell kinase (ITK) and tropomyosin receptor kinase A (TRKA) with an IC50 value of 1.0 nM and 96 % inhibition, respectively. | |||||||||||||||||||||
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Keywords
