3009018-61-2
3009018-61-2
Chemical Structure
σ1 Receptor/μ Opioid receptor modulator 2
- CAS No.: 3009018-61-2
- Formula:C23H31N3O
- Molecular Weight:365.51
InChIKey: PGTIFUTZJAGUST-UHFFFAOYSA-N
SMILES: O=C(N(C1=CC=CC=N1)CC(N2CCC(CC2)C3=CC=CC=C3)CC)CC
Biological Activity: σ1 Receptor/μ Opioid receptor modulator 2 (compound 4x) is a dual μOR agonist/σ1R antagonist, and displays picomolar μOR agonism activity (EC50: 0.6 ± 0.2 nM) and good σ1R inhibitory activity (Ki: 363.7 ± 5.6 nM). σ1 Receptor/μ Opioid receptor modulator 2 exhibits robust analgesic effects in various pain models[1].
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σ1 Receptor/μ Opioid receptor modulator 2 | σ1 Receptor/μ Opioid receptor modulator 2 (compound 4x) is a dual μOR agonist/σ1R antagonist, and displays picomolar μOR agonism activity (EC50: 0.6 ± 0.2 nM) and good σ1R inhibitory activity (Ki: 363.7 ± 5.6 nM). σ1 Receptor/μ Opioid receptor modulator 2 exhibits robust analgesic effects in various pain models. | |||||||||||||||||||||
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References
