2. GPCR/G Protein Neuronal Signaling
  3. Opioid Receptor Sigma Receptor
  4. σ1 Receptor/μ Opioid receptor modulator 2

σ1 Receptor/μ Opioid receptor modulator 2 

Cat. No.: HY-163065
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σ1 Receptor/μ Opioid receptor modulator 2 (compound 4x) is a dual μOR agonist/σ1R antagonist, and displays picomolar μOR agonism activity (EC50: 0.6 ± 0.2 nM) and good σ1R inhibitory activity (Ki: 363.7 ± 5.6 nM). σ1 Receptor/μ Opioid receptor modulator 2 exhibits robust analgesic effects in various pain models.

For research use only. We do not sell to patients.

σ1 Receptor/μ Opioid receptor modulator 2 Chemical Structure

σ1 Receptor/μ Opioid receptor modulator 2 Chemical Structure

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σ1 Receptor/μ Opioid receptor modulator 2 Related Antibodies

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Description

σ1 Receptor/μ Opioid receptor modulator 2 (compound 4x) is a dual μOR agonist/σ1R antagonist, and displays picomolar μOR agonism activity (EC50: 0.6 ± 0.2 nM) and good σ1R inhibitory activity (Ki: 363.7 ± 5.6 nM). σ1 Receptor/μ Opioid receptor modulator 2 exhibits robust analgesic effects in various pain models[1].

Molecular Weight

365.51

Formula

C23H31N3O
SMILES

O=C(N(C1=CC=CC=N1)CC(N2CCC(CC2)C3=CC=CC=C3)CC)CC
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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σ1 Receptor/μ Opioid receptor modulator 2 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

σ1 Receptor/μ Opioid receptor modulator 2Opioid ReceptorSigma Receptorpain modelsbifunctionalμOR/σ1RInhibitorinhibitorinhibit

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