σ1 Receptor/μ Opioid receptor modulator 2

σ1 Receptor/μ Opioid receptor modulator 2 (compound 4x) is a dual μOR agonist/σ1R antagonist, and displays picomolar μOR agonism activity (EC50: 0.6 ± 0.2 nM) and good σ1R inhibitory activity (Ki: 363.7 ± 5.6 nM). σ1 Receptor/μ Opioid receptor modulator 2 exhibits robust analgesic effects in various pain models.

For research use only. We do not sell to patients.

  • CAS No.: 3009018-61-2
  • Formula: C23H31N3O
  • Molecular Weight:365.51
  • Storage:

    Please store the product under the recommended conditions in the Certificate of Analysis.

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