3033060-62-4
3033060-62-4
Chemical Structure
LSD1-IN-15
- CAS No.: 3033060-62-4
- Formula:C22H20N2O
- Molecular Weight:328.41
IUPAC Name: N-(4-(2-aminocyclopropyl)phenyl)-3-(thiophen-2-yl)benzamide
InChIKey: SVQPTTBPYBICDV-UHFFFAOYSA-N
SMILES: NC1CC1C2=CC=C(C=C2)NC(C3=CC=CC(C4=CC=CC=C4)=C3)=O
Biological Activity: LSD1-IN-15 (compound 1b) is a potent LSD1 inhibitor. LSD1-IN-15 can inhibit LSD1-CoREST, MAO-A and MAO-B, with IC50 values of 0.149, 0.028, and 0.327 μM, respectively. LSD1-IN-15 displays cell growth arrest in prostate cancer LNCaP cells, with an IC50 of 9.9 μM[1].
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LSD1-IN-15 | LSD1-IN-15 (compound 1b) is a potent LSD1 inhibitor. LSD1-IN-15 can inhibit LSD1-CoREST, MAO-A and MAO-B, with IC50 values of 0.149, 0.028, and 0.327 μM, respectively. LSD1-IN-15 displays cell growth arrest in prostate cancer LNCaP cells, with an IC50 of 9.9 μM. | |||||||||||||||||||||
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References
Keywords
