359784-84-2
![[Ala17]-MCH Chemical Structure](http://file.medchemexpress.cn/product_pic/hy-p1204.gif "[Ala17]-MCH Chemical Structure")
Chemical Structure
[Ala17]-MCH
- CAS No.: 359784-84-2
- Formula:C97H155N29O26S4
- Molecular Weight:2271.71
IUPAC Name: (6S,9S,12S,15S,18S,21S)-1,21-diamino-6-(((3R,8R,11S,14S,20S,23S,26S,29S)-3-(((S)-1-(((S)-5-amino-1-(((S)-1-carboxy-2-methylpropyl)amino)-1,5-dioxopentan-2-yl)amino)-1-oxopropan-2-yl)carbamoyl)-20,29-bis(3-guanidinopropyl)-26-(4-hydroxybenzyl)-14-isobutyl-
InChIKey: IVEALEKXBDDRGB-VWUJWYMQSA-N
SMILES: O=C1N2C(CCC2)([H])C(N[C@@H](CSSC[C@@H](C(N[C@H](C(N[C@H](C(NCC(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H]1CCCNC(N)=N)=O)CC3=CC=C(C=C3)O)=O)C(C)C)=O)CCCNC(N)=N)=O)=O)CC(C)C)=O)CCSC)=O)NC([C@H](CCCNC(N)=N)NC([C@H](CC(C)C)NC([C@H](CCSC)NC([C@H](CC(O)=O)NC([C@@H](NC([C@@H](N)CC(O)=O)=O)CC4=CC=CC=C4)=O)=O)=O)=O)=O)C(N[C@@H](C)C(N[C@@H](CCC(N)=O)C(N[C@H](C(O)=O)C(C)C)=O)=O)=O)=O
Biological Activity: [Ala17]-MCH, a MCH analogue (HY-P1525A), is a selective ligand for MCHR1 (Ki=0.16 nM) over MCHR2 (Ki=34 nM). [Eu3+ chelate-labeled [Ala17]-MCH shows high affnity for MCHR1 (Kd=0.37 nM) while has little demonstrable binding affnity for MCHR2[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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[Ala17]-MCH | 98.28% | [Ala17]-MCH, a MCH analogue (HY-P1525A), is a selective ligand for MCHR1 (Ki=0.16 nM) over MCHR2 (Ki=34 nM). [Eu3+ chelate-labeled [Ala17]-MCH shows high affnity for MCHR1 (Kd=0.37 nM) while has little demonstrable binding affnity for MCHR2. | ||||||||||||||||||||
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Keywords
